Olaparib | CAS#763113-22-0 MedChemExpress(MCE)貨號HY-10162

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MCE (MedChem Express) Olaparib
MCE總部位於美國新澤西,提供種類齊全的化學及生化研究用產品,包括創新的生命科學試劑,reference compounds(標準化合物),APIs(原料藥)及Natural compounds(天然化合物)以提供實驗室或科學研究之用,MedChemExpress(MCE)產品50000+ 特異性抑制劑、化合物庫、重組蛋白,專注於信號通路和疾病研究領域。全球文獻廣泛引用,質控體系嚴格,品質100%
CAS No. : 763113-22-0
Olaparib (AZD2281; KU0059436) | CAS#763113-22-0 MedChemExpress(MCE)貨號HY-10162
AZD2281; KU0059436
Olaparib (AZD2281; KU0059436) 是一種有效的口服活性 PARP 抑制劑,對 PARP1 和 PARP2 的 IC50 分別為 5 和 1 nM。 Olaparib 是一種自噬(autophagy )和線粒體自噬激活劑(mitophagy activator)。
Olaparib purchased from MCE. Usage Cited in: Oncogene. 2018 Jan 18;37(3):341-351. [Abstract]
PTEN-deficient endometrioid endometrial cancer cell lines are treated with drugs as indicated for 24 h. Phosphorylated AKT, S6RP and 4EBP1 proteins and cleaved PARP are detected by western blot. Vinculin served as a loading control.
Olaparib purchased from MCE. Usage Cited in: Gynecol Oncol. 2019 Jan;152(1):157-165. [Abstract]
Immunohistochemistry of RAD51 and γ-H2AX in samples of SKOV3 tumors. Representative sections are taken from tumor tissue of control, scrambled shRNA treated, Olaparib + scrambled shRNA treated, or Olaparib + CCND1-shRNA treated mice.
Olaparib purchased from MCE. Usage Cited in: J Biomed Sci. 2019 Feb 4;26(1):14. [Abstract]
Inhibition of NFBD1 results in defective γ-H2AX foci formation after Olaparib exposure, cells are exposed to Olaparib for 24 h, and the γ-H2AX positive cells are determined by FCM
MedChemexpress (MCE) 產品
MCE (MedChemexpress) 總部位於美國新澤西,提供種類齊全的化學及生化研究用產品,包括創新的生命科學試劑,reference compounds (標準化合物),APIs (原料藥) 及Natural compounds (天然化合物)以提供實驗室或科學研究之用,MedChemExpress(MCE)產品50000+ 特異性抑制劑、化合物庫、重組蛋白,專注於信號通路和疾病研究領域。全球文獻廣泛引用,質控體系嚴格,品質100%。官網連結 https://www.medchemexpress.com
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