Avasimibe ACAT抑制劑 | cholesterol acyltransferase Inhibitors 貨號: 9506-25

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特點
ACAT Inhibitors | Avasimibe抑制劑 | 貨號: 9506-25 An acyl coenzyme A: cholesterol acyltransferase (ACAT) inhibitor
Avasimibe是口服生物抑製劑:acyl coenzyme A inhibitor;膽固醇酰基轉移酶(ACAT) (IC₅₀ = 60 nM)。Avasimibe亦是抑制主要藥物代謝酶CYP2C9 (IC₅₀ = 2.9 µM ), CYP1A2 (IC₅₀ = 13.9 µM), and CYP2C19 (IC₅₀ = 26.5 µM)。
Molecular Formula: C₂₉H₄₃NO₄S
Molecular Weight: 501.7
Purity: ≥98% by HPLC
Solubility:DMSO (>35 mg/ml)
| Catalog # | Product Name+ | Size |
| 9506-5 | Avasimibe | 5 mg |
| 9506-25 | Avasimibe | 25 mg |
| 2053-1 | Pellitorine | 1 mg |
| 2053-5 | Pellitorine | 5 mg |
| 2214-250 | Terpendole C | 250 µg |
| 2214-1000 | Terpendole C | 1 mg |

