CP-640186抑制劑 |混合型ACC Inhibitors Biovision貨號: 9422-25

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混合型ACC Inhibitors | CP-640186抑制劑 | 貨號: 9422-25
A mixed ACC (Acetyl-CoA carboxylase) inhibitor
CP-640186是混合型ACC(乙酰輔酶A羧化酶)抑制劑(ACC-1 IC 50= 53納米; ACC-2 IC 50=61納米),降低malonyl–CoA水平,在體外和體內實驗中,抑制肝脂肪酸和甘油三酯的合成,以及刺激肌肉脂肪酸氧化及降低大鼠body RQ。CP-640186 is a mixed ACC (Acetyl-CoA carboxylase) inhibitor (ACC-1 IC₅₀ = 53 nM; ACC-2 IC₅₀ = 61 nM) that lowers malonyl-CoA levels and inhibits hepatic fatty acid and triglyceride synthesis in vitro and in vivo, as well as stimulates muscle fatty acid oxidation and lowers whole body RQ in rats.
Molecular Formula: C₃₀H₃₅N₃O₃
Molecular Weight: 485.62
Purity: ≥98% by HPLC
Solubility: DMSO
| Catalog # | Product Name+ | Size |
| 1717-5 | ACC2 Inhibitor | 5 mg |
| 1717-1 | ACC2 Inhibitor | 1 mg |
| 9422-5 | CP-640186 | 5 mg |
| 9422-25 | CP-640186 | 25 mg |
更多酵素型抑制劑商品: ACE抑制劑類 | AR抑制劑類 | AKR抑制劑類 | adenylyl cyclase 抑制劑類 | AAC抑制劑 | ACAT抑制劑

