【G 418 sulfate (80 S 核醣體延伸抑制劑) 】 CAS# 108321-42-2 APExBIO貨號A2513
雷帕黴菌（Rapamycin）| Romidepsin (FK228, depsipeptide) | Daptomycin | G-418 (80 S 核醣體延伸抑制劑)
G-418 (80 S 核醣體延伸抑制劑) | CAS# 108321-42-2 APExBIO貨號A2513
G-418 is an elongation inhibitor of 80 S ribosomes [1].
G-418 是 80 S 核醣體(80 S ribosomes)的延伸抑制劑(elongation inhibitor)。
產品介紹G418是一種氨基糖苷類抗生素(aminoglycoside antibiotic)，具有廣譜活性(wide spectrum of activity)，對細菌(bacteria)、酵母菌(yeasts)、真菌(fungi)、藻類(algae)、植物(plant)甚至動物細胞(animal cells)都有活性。 G418 通常用作原核和真核生物(eukaryotes)中的克隆(cloning selection)選擇，濃度為 1 至 300ug/ml。在細菌臨床分離株的抗生素耐藥性研究中，發現所有攜帶3′-O-氨基糖苷磷酸轉移酶(3′-O-aminoglycoside phosphotransferases)的菌株均對G418耐藥。在這些磷酸轉移酶中，I 型和 II 型分別由轉座因子 TnS 和 Tn601 編碼 [2]。
除了選擇功能(selector function)外，還發現 G418 對牛病毒性腹瀉病毒 (bovine viral diarrhea virus , BVDV) 具有抗病毒活性。 G418 以劑量依賴性方式防止 DENV-2 感染 BHK 細胞引起的細胞病變效應 (CPE)，EC50 值為 3±0.4 g/ml [3]。
| Physical Appearance | A solid |
| Storage | Store at -20°C |
| M.Wt | 692.71 |
| Cas No. | 108321-42-2 |
| Formula | C20H40N4O10·2H2SO4 |
| Synonyms | Antibiotic G418 |
| Solubility | insoluble in EtOH; insoluble in DMSO; ≥64.6 mg/mL in H2O |
| Chemical Name | 2-[4,6-diamino-3-[3-amino-4,5-dihydroxy-6-(1-hydroxyethyl)oxan-2-yl]oxy-2-hydroxycyclohexyl]oxy-5-methyl-4-(methylamino)oxane-3,5-diol;sulfuric acid |
| SDF | Download SDF |
| Canonical SMILES | CC(C1C(C(C(C(O1)OC2C(CC(C(C2O)OC3C(C(C(CO3)(C)O)NC)O)N)N)N)O)O)O.OS(=O)(=O)O.OS(=O)(=O)O |
| Shipping Condition | Ship with blue ice, or upon other requests. |
| General tips | For obtaining a higher solubility, please warm the tube at 37°C and shake it in the ultrasonic bath for a while. We do not recommend long-term storage for the solution, please use it up soon. |
產品引用
- 1. Zhang C, Duan Y, et al. “TFEB mediates immune evasion and resistance to mTOR inhibition of renal cell carcinoma via induction of PD-L1.” Clin Cancer Res. 2019 Aug 5. pii: clincanres.0733.2019. PMID:31383732
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| A3222 | Baricitinib phosphate | 1187595-84-1 | 99.59% | JAK1/JAK2 inhibitor |
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| A3268 | CAL-130 Hydrochloride | 1431697-78-7 | 98.00% | PI3K inhibitor |
| A3270 | Calcifediol monohydrate | 63283-36-3 | 99.43% | Prehormone;vitamin D3 metabolite |
| A3271 | Calcipotriol | 112965-21-6 | 98.00% | Vitamin D3 analog,regulates cell differentiation and proliferation |
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| A3335 | Curcumin | 458-37-7 | 98.36% | Tyrosinase inhibitor |
| A3336 | CVT-313 | 199986-75-9 | 98.04% | Cdk2 inhibitor |
| A3337 | CX-6258 | 1202916-90-2 | 98.28% | Pan-Pim kinases Inhibitor |
| A3339 | CYT387 sulfate salt | 1056636-06-6 | 98.00% | JAK1/JAK2 inhibitor |
| A3340 | CZC24832 | 1159824-67-5 | 98.00% | Selective PI3K-γ inhibitor |
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| A3346 | Dabigatran ethyl ester | 429658-95-7 | 98.00% | Thrombin activity inhibitor |
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| A3366 | Dipraglurant | 872363-17-2 | 98.00% | mGluR5 antagonist |
| A3368 | DMAT | 749234-11-5 | 98.60% | CK2 inhibitor,potent and selective |
| A3369 | DMP 777 | 157341-41-8 | 98.00% | Leukocyte elastase (HLE) inhibitor |
| A3370 | Docetaxel Trihydrate | 148408-66-6 | 99.78% | Depolymerisation of microtubules inhibitor |
| A3371 | Doramectin | 117704-25-3 | 97.08% | Antiparasitic antibiotic |
| A3374 | Dronedarone | 141626-36-0 | 99.58% | CYP3A4 and 2D6 inhibitor,moderate |
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| A3378 | E-3810 | 1058137-23-7 | 98.00% | VEGF/FGF dual inhibitor, potent and selective |
| A3380 | Ebrotidine | 100981-43-9 | 98.00% | H2-receptor antagonist,competitive |
| A3381 | Edoxaban | 480449-70-5 | 99.27% | Factor Xa inhibitor |
| A3383 | Edoxaban tosylate monohydrate | 1229194-11-9 | 99.34% | Oral factor Xa inhibitor |
| A3384 | Elacridar | 143664-11-3 | 98.17% | BCRP inhibitor |
| A3385 | Elacridar hydrochloride | 143851-98-3 | 98.00% | BCRP and P-GP inhibitor |
| A3387 | Eltrombopag Olamine | 496775-62-3 | 98.49% | C-mpl agonist |
| A3389 | EMD638683 | 1181770-72-8 | 98.46% | SGK1 inhibitor |
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| A3394 | Epothilone D | 189453-10-9 | 98.00% | Natural polyketide compound |
| A3395 | Ercalcidiol | 21343-40-8 | 98.00% | Vitamin D2 metabolite,ligand of VDR-like receptors |
| A3396 | Ercalcitriol | 60133-18-8 | 98.00% | Active metabolite of vitamin D2 |
| A3397 | Erlotinib | 183321-74-6 | 99.47% | EGFR tyrosine kinase inhibitor |
| A3399 | Esomeprazole Magnesium trihydrate | 217087-09-7 | 98.32% | Proton pump inhibitor |
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| A3403 | Etofenamate | 30544-47-9 | 98.05% | Non-steroidal anti-inflammatory drug |
| A3404 | Etomoxir | 124083-20-1 | 99.75% | (CPT)-1 and DGAT activity inhibitor |
| A3405 | Etoricoxib | 202409-33-4 | 99.82% | Specific COX-2 inhibitor |
| A3407 | EVP-6124 hydrochloride | 550999-74-1 | 99.85% | Alpha7 nAChR agonist |
| A3408 | Exendin-4 | 141758-74-9 | 99.66% | GLP-1 activator |
| A3411 | Faropenem daloxate | 141702-36-5 | 98.00% | Oral penem,beta-lactam antibiotic |
| A3412 | Fenretinide | 65646-68-6 | 98.00% | Synthetic retinoid agonist |
| A3413 | FH535 | 108409-83-2 | 99.62% | Wnt/B-catenin inhibitor |
| A3415 | Firategrast | 402567-16-2 | 99.56% | α4β1/α4β7 integrin antagonist |
| A3416 | FK 3311 | 116686-15-8 | 98.00% | Selective COX-2 inhibitor |
| A3417 | Flavopiridol | 146426-40-6 | 99.52% | Pan-cdk inhibitor |
| A3418 | Flecainide acetate | 54143-56-5 | 99.82% | Antiarrhythmic drug |
| A3419 | Fluvastatin | 93957-54-1 | 98.33% | HMGCR inhibitor |
| A3420 | FMK | 821794-92-7 | 98.82% | RSK inhibitor |
| A3421 | Fosamprenavir Calcium Salt | 226700-81-8 | 99.71% | Prodrug of antiretroviral protease inhibitor amprenavir |
| A3423 | Galanthamine | 357-70-0 | 99.12% | Acetylcholinesterase inhibitor |
| A3424 | Gambogic Acid | 2752-65-0 | 98.54% | Caspase activator and apoptosis inducer |
| A3429 | GANT 58 | 64048-12-0 | 99.38% | GLI antagonist,novel and potent |
| A3432 | GDC-0941 dimethanesulfonate | 957054-33-0 | 99.78% | PI3K inhibitor |
| A3433 | Gefitinib hydrochloride | 184475-55-6 | 99.87% | Potent EGFR inhibitor |
| A3434 | Genz-644282 | 529488-28-6 | 98.00% | Non-camptothecin inhibitor of topoisomerase I |
| A3435 | glucagon receptor antagonists 1 | 503559-84-0 | 98.00% | Glucagon receptor antagonist,highly potent |
| A3436 | glucagon receptor antagonists 2 | 202917-18-8 | 98.00% | Glucagon receptor antagonist,highly potent |
| A3437 | glucagon receptor antagonists 3 | 202917-17-7 | 98.00% | Glucagon receptor antagonist |
| A3438 | Glucocorticoid receptor agonist | 1245526-82-2 | 98.00% | Glucagon receptor antagonist |
| A3440 | Glyoxalase I inhibitor | 221174-33-0 | 98.00% | Glyoxalase I inhibitor |
| A3441 | GPR120 modulator 1 | 1050506-75-6 | 98.00% | GPR120 modulator |
| A3442 | GPR120 modulator 2 | 1050506-87-0 | 98.00% | GPR120 modulator |
| A3443 | Granisetron | 109889-09-0 | 98.00% | Serotonin 5-HT3 receptor antagonist |
| A3444 | GS-9620 | 1228585-88-3 | 98.01% | TLR-7 agonist |
| A3445 | GSK 525768A | 1260530-25-3 | 98.00% | inactive stereoisomer of I-BET-762 |
| A3446 | GSK126 | 1346574-57-9 | 98.32% | EZH2 inhibitor |
| A3448 | GSK2606414 | 1337531-36-8 | 98.18% | PERK inhibitor,potent and selective |
| A3449 | GSK343 | 1346704-33-3 | 98.95% | EZH2 inhibitor,potent,selective and cell permeable |
| A3450 | GSK-923295 | 1088965-37-0 | 98.28% | CENP-E inhibitor,small-molecule |
| A3451 | Guanfacine hydrochloride | 29110-48-3 | 99.41% | α2A-adrenoceptor agonist |
| A3452 | GW-1100 | 306974-70-9 | 98.00% | GPR40 antagonist |
| A3453 | GW1929 | 196808-24-9 | 98.00% | Potent PPARγ agonist |
| A3454 | GW3965 | 405911-09-3 | 98.00% | HLXRα/hLXRβ agonist,potent and selective |
| A3456 | GW843682X | 660868-91-7 | 98.00% | PLK1/PLK3 inhibitor,potent and selective |
| A3460 | HhAntag | 496794-70-8 | 98.95% | GLI1-mediated transcription inhibitor |
| A3461 | HIV-1 integrase inhibitor | 544467-07-4 | 98.00% | Uesful for anti-HIV |
| A3465 | HOE 33187 | 23623-08-7 | 98.00% | Blue fluorescent dyes |
| A3466 | Hoechst 33258 | 23491-45-4 | 99.88% | Blue fluorescent dyes |
| A3472 | Hoechst 33342 | 875756-97-1 | 98.84% | Blue fluorescent dyes |