單胺氧化酶B高通量篩選分析套組| Monoamine Oxidase B (MAO-B) Inhibitor Screening Kit (Fluorometric) 貨號K797

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商品: Monoamine Oxidase B (MAO-B) Inhibitor Screening Kit (Fluorometric) 單胺氧化酶B高通量篩選分析套組
產品規格: 胺氧化酶B高通量篩選分析套組 貨號K797 | 100個分析 Monoamine Oxidase B (MAO-B) Inhibitor Screening Kit (Fluorometric)
產品描述: Monoamine oxidases單胺氧化酶(MAO,EC 1.4.3.4)是可以氧化多種內源性伯胺的酶家族。以它們的substrate底物,inhibitor specificity抑制特異性和tissue localization組織定位;鑑定了兩種同種型,MAO-A和MAO-B。MAO-B可以氧化伯胺,但是與MAO-A相比,其特定底物(即芐胺,苯乙胺)的列表更有限。 MAO-B是線粒體結合的酶,其在整個腦和其他組織中普遍表達。已經在包括帕金森病,阿爾茨海默氏病和煙草成癮的許多研究中進行了研究。特異性MAO-B抑制劑如司來吉蘭和雷沙吉蘭已經用於治療帕金森病患者,但它們的益處被認為相當溫和。 BioVision的MAO-B抑制劑篩選試劑盒提供了快速,簡單,靈敏和可靠的測試,適用於高通量篩選MAO-B抑制劑。該測定基於H 2 O 2的螢光檢測,H 2 O 2是MAO底物的氧化脫氨期間產生的副產物之一。

| Size | 100 assays |
| SKU+Size | K797-100 |
| Detection Method | Fluorescence (Ex/Em = 535/587 nm) |
| Applications | Screening/studying/characterizing MAO-B inhibitors |
| Features & Benefits | • Rapid & sensitive • High-throughput assay to screen/study/characterize potential inhibitors of monoamine oxidase B • Includes Inhibitor Control [Selegiline] |
| Kit Components | • MAO-B Assay Buffer • OxiRed™ Probe (in DMSO) • MAO-B Enzyme (Lyophilized) • MAO-B Substrate (Lyophilized) • Developer (Lyophilized) • Inhibitor Control (Clorgyline) (Lyophilized) |
