{"id":34208,"date":"2022-09-16T16:42:16","date_gmt":"2022-09-16T08:42:16","guid":{"rendered":"http:\/\/biopioneer.com.tw\/?p=34208"},"modified":"2025-11-15T15:30:07","modified_gmt":"2025-11-15T07:30:07","slug":"ampicillin-sodium-cas-69-52-3-apexbio-%e8%b2%a8%e8%99%9fa2510","status":"publish","type":"post","link":"https:\/\/biopioneer.com.tw\/?p=34208","title":{"rendered":"\u5b89\u6bd4\u897f\u6797Ampicillin sodium | CAS# 69-52-3 APExBIO  \u8ca8\u865fA2510"},"content":{"rendered":"<p><strong><span style=\"font-size: 12pt; color: #ff6600;\"><span style=\"font-size: 14pt;\"><span style=\"color: #800080;\">\u03b2-\u5167\u91af\u80fa\u985e\u6297\u751f\u7d20\u7cfb\u5217\u5546\u54c1-&gt;&gt;<\/span><\/span><span style=\"font-size: 14pt;\">\u5b89\u6bd4\u897f\u6797Ampicillin sodium<\/span><\/span><\/strong><\/p>\n<p>APExBIO Technology LLC \u662f\u4e00\u5bb6\u9818\u5148\u7684\u5c0f\u5206\u5b50\u6291\u5236\u5291 (Small Molecule Inhibitors)\/\u6d3b\u5316\u5291(Activators)\u3001\u5316\u5408\u7269\u5eab( Compound Libraries)\u3001\u80dc\u80bd(Peptides)\u3001\u6aa2\u6e2c\u8a66\u5291\u76d2(Assay Kits)\u3001\u87a2\u5149\u6a19\u8a18(Fluorescent Label)\u3001\u9176(Enzymes)\u3001\u4fee\u98fe\u6838\u82f7\u9178(Modified Nucleotides)\u3001mRNA \u5408\u6210\u4ee5\u53ca\u5404\u7a2e\u5206\u5b50\u751f\u7269\u5b78\u5de5\u5177\u7684\u4f9b\u61c9\u5546\u3002APExBIO\u63d0\u4f9b\u5ee3\u6cdb\u7684\u7522\u54c1\u7dda\uff0c\u6db5\u84cb 20 \u591a\u500b\u4e0d\u540c\u7684\u7814\u7a76\u9818\u57df\uff0c\u4f8b\u5982\u764c\u75c7(cancer)\u3001\u514d\u75ab\u5b78(immunology)\u3001\u795e\u7d93\u79d1\u5b78(neurosciences)\u3001\u7d30\u80de\u51cb\u4ea1(apoptosis)\u548c\u8868\u89c0\u907a\u50b3\u5b78(epigenetics)\u7b49\u3002\u516c\u53f8\u7e3d\u90e8\u4f4d\u65bc\u7f8e\u570b\u5fb7\u5dde\u4f11\u58eb\u9813USA (Houston, Texas)\uff0c\u81f4\u529b\u65bc\u670d\u52d9\u5168\u7403\u5ba2\u6236\u3002\u9ad8\u5ea6\u91cd\u8996\u7522\u54c1\u54c1\u8cea\u3002\u6240\u6709\u7522\u54c1\u5747\u9075\u5faa\u56b4\u683c\u7684\u751f\u7522\u6307\u5357\uff0c\u4e26\u9644\u6709\u5206\u6790\u8b49\u66f8\u3001HPLC\u3001\u8cea\u8b5c(Mass Spectrum)\u548cHMNR\u4ee5\u53ca\u9ad4\u5916\u9a57\u8b49(in vitro validation)\u3002 APExBIO\u7522\u54c1\u5df2\u88ab\u300aNature\u300b\u3001\u300aCell\u300b\u548c\u300aScience\u300b\u7b49\u773e\u591a\u9802\u7d1a\u540c\u884c\u8a55\u5be9\u671f\u520a\u5f15\u7528\u3002<a href=\"https:\/\/biopioneer.com.tw\/?news=apexbio%e5%8f%b0%e7%81%a3%e4%bb%a3%e7%90%86%e5%95%86-brandagency%e4%bb%a3%e7%90%86%e5%93%81%e7%89%8c-apexbio-2\"><span style=\"color: #ff0000;\"><em><strong><span style=\"text-decoration: underline;\">&gt;&gt;\u66f4\u591aAPExBio\u5546\u54c1<\/span><\/strong><\/em><\/span><\/a><\/p>\n<p><img decoding=\"async\" loading=\"lazy\" class=\"\" src=\"https:\/\/biopioneer.com.tw\/wp-content\/uploads\/downloads\/2025\/06\/%E5%A4%AA%E9%BC%8E-APExBIO-Technology-LLC-%E5%93%81%E7%89%8C.png\" width=\"1099\" height=\"274\" \/><\/p>\n<p><span style=\"color: #00ccff;\"><a style=\"color: #00ccff;\" href=\"http:\/\/biopioneer.com.tw\/?p=34208\"><strong><span style=\"color: #33cccc; font-size: 12pt;\">\u5b89\u6bd4\u897f\u6797Ampicillin sodium | CAS# 69-52-3 APExBIO\u00a0 \u8ca8\u865fA2510<\/span><\/strong><\/a><\/span><\/p>\n<p><img decoding=\"async\" src=\"http:\/\/biopioneer.com.tw\/wp-content\/uploads\/2022\/09\/Ampicillin-sodium-CAS-69-52-3-APExBIO-%E8%B2%A8%E8%99%9FA2510-300x281.png\" alt=\"Ampicillin sodium CAS# 69-52-3 APExBIO \u8ca8\u865fA2510\" \/><\/p>\n<p>Ampicillin sodium is a competitive inhibitor of the enzyme transpeptidase with IC50 value of 1.8 \u03bcg\/ml [1].<\/p>\n<p>\u5b89\u6bd4\u897f\u6797(Ampicillin)\u662f\u4e00\u7a2e\u9176\u8f49\u80bd\u9176\u7684\u7af6\u722d\u6027\u6291\u5236\u5291\uff0cIC50 \u503c\u70ba 1.8 \u03bcg\/ml [1]\u3002<\/p>\n<p>\u5b89\u6bd4\u897f\u6797(Ampicillin)\u662f\u4e00\u7a2e\u03b2-\u5167\u91af\u80fa\u985e\u6297\u751f\u7d20(\u03b2-lactam antibiotic)\uff0c\u901a\u904e\u6291\u5236\u8f49\u80bd\u9176\u53cd\u61c9(transpeptidase reactions)\u4f86\u6bba\u6b7b\u7d30\u83cc\u3002\u8f49\u80bd\u9176(Transpeptidase)\u53c3\u8207\u7d30\u80de\u58c1\u751f\u7269\u5408\u6210(cell wall biosynthesis)\u7684\u6700\u5f8c\u968e\u6bb5\uff0c\u5c0d\u5176\u7684\u6291\u5236\u6700\u7d42\u5c0e\u81f4\u7d30\u80de\u88c2\u89e3(cell lysis) [1]\u3002\u5728\u4e59\u919a\u8655\u7406\u7684\u5927\u8178\u687f\u83cc146\u7d30\u80de\u4e2d\uff0c\u5b89\u6bd4\u897f\u6797(Ampicillin)\u5728\u4f4e\u65bc0.5 \u03bcg\/ml\u7684\u6fc3\u5ea6\u4e0b\u5c0d\u8f49\u80bd\u9176\u53cd\u61c9(transpeptidase reaction)\u6c92\u6709\u660e\u986f\u7684\u6291\u5236\u4f5c\u7528\uff0c\u4f46\u57281.8 \u03bcg\/ml\u7684\u6fc3\u5ea6\u4e0b\u8868\u73fe\u51fa50%\u7684\u6291\u5236\u4f5c\u7528\u3002\u5728\u5927\u8178\u687f\u83cc 146 \u7d30\u80de\u4e2d\uff0c\u5b89\u6bd4\u897f\u6797(Ampicillin)\u7684\u6700\u4f4e\u6291\u83cc\u6fc3\u5ea6 (MIC) \u70ba 3.1 \u03bcg\/ml [1]\u3002\u5728\u5927\u8178\u687f\u83cc(<em>E. coli)<\/em>\u548c\u50b7\u5bd2\u6c99\u9580\u6c0f\u83cc\u4e2d\uff0c\u6fc3\u5ea6\u63a5\u8fd1 MIC \u503c\u7684\u5b89\u6bd4\u897f\u6797(Ampicillin)\u548c Epicillin \u6bba\u6b7b\u7d30\u83cc\u7684\u901f\u5ea6\u6bd4\u963f\u83ab\u897f\u6797\u6162 [2]\u3002\u5728\u5be6\u9a57\u6027\u5c0f\u9f20\u611f\u67d3\u4e2d\uff0c\u4ee5 0.2 ml\/20 g \u7684\u5291\u91cf\u53e3\u670d\u6216\u76ae\u4e0b\u6ce8\u5c04\u5b89\u6bd4\u897f\u6797(Ampicillin)\u5c0d\u5927\u591a\u6578\u611f\u67d3\u7684\u6cbb\u7642\u6548\u679c\u660e\u986f\u512a\u65bc Epicillin \u548c Amoxycillin [2]\u3002<\/p>\n<table width=\"1128\">\n<tbody>\n<tr>\n<td>Storage<\/td>\n<td>Store at -20\u00b0C<\/td>\n<\/tr>\n<tr>\n<td>M.Wt<\/td>\n<td>371.4<\/td>\n<\/tr>\n<tr>\n<td>Cas No.<\/td>\n<td>69-52-3<\/td>\n<\/tr>\n<tr>\n<td>Formula<\/td>\n<td>C<sub>16<\/sub>H<sub>18<\/sub>N<sub>3<\/sub>NaO<sub>4<\/sub>S<\/td>\n<\/tr>\n<tr>\n<td>Solubility<\/td>\n<td>\u226518.57 mg\/mL in H2O; \u226573.6 mg\/mL in DMSO; \u226575.2 mg\/mL in EtOH<\/td>\n<\/tr>\n<tr>\n<td>Chemical Name<\/td>\n<td>sodium;(2S,5R,6R)-6-[[(2R)-2-amino-2-phenylacetyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylate<\/td>\n<\/tr>\n<tr>\n<td>SDF<\/td>\n<td><a href=\"https:\/\/www.apexbt.com\/downloader\/sdf\/A2510.sdf\">Download SDF<\/a><\/td>\n<\/tr>\n<tr>\n<td>Canonical SMILES<\/td>\n<td>CC1(C(N2C(S1)C(C2=O)NC(=O)C(C3=CC=CC=C3)N)C(=O)[O-])C.[Na+]<\/td>\n<\/tr>\n<tr>\n<td>Shipping Condition<\/td>\n<td>Ship with blue ice, or upon other requests.<\/td>\n<\/tr>\n<tr>\n<td>General tips<\/td>\n<td>For obtaining a higher solubility, please warm the tube at 37\u00b0C and shake it in the ultrasonic bath for a while. We do not recommend long-term storage for the solution, please use it up soon.<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<p><img decoding=\"async\" loading=\"lazy\" class=\"\" src=\"http:\/\/biopioneer.com.tw\/wp-content\/uploads\/2022\/12\/%E5%93%81%E7%89%8C%E7%B9%AA%E5%9C%96-Apexbio_%E5%B7%A5%E4%BD%9C%E5%8D%80%E5%9F%9F-1-300x300.jpg\" width=\"203\" height=\"225\" \/><\/p>\n<p><a href=\"http:\/\/www.apexbt.com\/\"><span style=\"font-size: 14pt; color: #ff6600;\"><strong><span style=\"color: #800080;\"><span style=\"font-size: 14pt;\">APExBIO\u53f0\u7063\u4ee3\u7406\u5546:\u00a0 <\/span><\/span><\/strong><\/span><\/a><span style=\"font-size: 14pt;\"><a href=\"https:\/\/www.apexbt.com\/\"><span style=\"color: #ff99cc;\"><span style=\"color: #ff6600;\">https:\/\/www.apexbt.com\/<\/span><\/span><\/a><\/span><\/p>\n<p>APExBIO\u63d0\u4f9b\u512a\u8cea\u7684\u80dc\u80bd\u548c\u751f\u7269\u5206\u6790\u8a66\u5291\uff0c\u5ee3\u6cdb\u7522\u54c1\u7dda\u5982Protease\u3001Chromatin\/Epigenetics\u8868\u89c0\u907a\u50b3\u5b78\u3001MAPK Signal\u3001DNA Damege\/DNA repair\u3001\u7d30\u80de\u51cb\u4ea1\u3001\u816b\u7624\u751f\u7269\u5b78\u3001Stem cell\u7b49\u7814\u7a76\u9818\u57df\uff0c \u9084\u63d0\u4f9b\u5b9a\u5236\u7684\u670d\u52d9\uff0c\u5305\u62ec\u591a\u80bd\u5408\u6210\uff0c\u6297\u9ad4\u7684\u751f\u7522\u548c\u6aa2\u6e2c\u7684\u767c\u5c55\u3002\u7522\u54c1\u7ddaDNA\/RNA prep kit\u3001Drug Screening panel\u3001Bioactive peptides\u3001Growth factors\u3001Biotinylation Reagents\u3001tag peptides\u3001amino Acids\u3001Growth factors\u7b49\u3002APExBIO\u7522\u54c1\u8cea\u91cf\u90fd\u4f34\u96a8\u8457\u8b49\u66f8\u7684\u5206\u6790\uff0c\u9ad8\u6548\u6db2\u76f8\u8272\u8b5c\uff0c\u8cea\u8b5c\uff0c\u548cHMNR\u6578\u64da\u3002<\/p>\n<p><img decoding=\"async\" loading=\"lazy\" class=\"\" src=\"http:\/\/biopioneer.com.tw\/wp-content\/uploads\/2024\/09\/line-2_%E5%B7%A5%E4%BD%9C%E5%8D%80%E5%9F%9F-1.jpg\" width=\"302\" height=\"230\" \/><\/p>\n<table style=\"height: 2756px;\" width=\"1152\">\n<tbody>\n<tr>\n<td width=\"62\">Cat#<\/td>\n<td width=\"313\">Product Name<\/td>\n<\/tr>\n<tr>\n<td>A8743<\/td>\n<td>SYBR Safe DNA Gel Stain<\/td>\n<\/tr>\n<tr>\n<td>A6001<\/td>\n<td>3X (DYKDDDDK) Peptide<\/td>\n<\/tr>\n<tr>\n<td>K1018<\/td>\n<td>Cell Counting Kit-8 (CCK-8)<\/td>\n<\/tr>\n<tr>\n<td>A1902<\/td>\n<td>Z-VAD-FMK<\/td>\n<\/tr>\n<tr>\n<td>A3008<\/td>\n<td>Y-27632 dihydrochloride<\/td>\n<\/tr>\n<tr>\n<td>A6002<\/td>\n<td>DYKDDDDK tag Peptide<\/td>\n<\/tr>\n<tr>\n<td>B8362<\/td>\n<td>2&#8217;3&#8242;-cGAMP (sodium salt)<\/td>\n<\/tr>\n<tr>\n<td>F4002<\/td>\n<td>Phos binding reagent (Phosbind) acrylamide<\/td>\n<\/tr>\n<tr>\n<td>A8011<\/td>\n<td>Biotin-tyramide<\/td>\n<\/tr>\n<tr>\n<td>A2585<\/td>\n<td>MG-132<\/td>\n<\/tr>\n<tr>\n<td>F4005<\/td>\n<td>Prestained Protein Marker (Triple color, EDTA free, 10-250 kDa)<\/td>\n<\/tr>\n<tr>\n<td>B1274<\/td>\n<td>AP20187<\/td>\n<\/tr>\n<tr>\n<td>K1007<\/td>\n<td>Protease Inhibitor Cocktail(EDTA-Free,100X in DMSO)<\/td>\n<\/tr>\n<tr>\n<td>B8226<\/td>\n<td>InstaBlue Protein Stain Solution<\/td>\n<\/tr>\n<tr>\n<td>A3011<\/td>\n<td>CHIR-99021 (CT99021)<\/td>\n<\/tr>\n<tr>\n<td>A3007<\/td>\n<td>ABT-263 (Navitoclax)<\/td>\n<\/tr>\n<tr>\n<td>B1524<\/td>\n<td>Erastin<\/td>\n<\/tr>\n<tr>\n<td>B6055<\/td>\n<td>TCEP hydrochloride<\/td>\n<\/tr>\n<tr>\n<td>K1031<\/td>\n<td>Phusion high-fidelity DNA polymerase<\/td>\n<\/tr>\n<tr>\n<td>B1387<\/td>\n<td>(-)-Blebbistatin<\/td>\n<\/tr>\n<tr>\n<td>B4664<\/td>\n<td>T-5224<\/td>\n<\/tr>\n<tr>\n<td>A8183<\/td>\n<td>Trichostatin A (TSA)<\/td>\n<\/tr>\n<tr>\n<td>B3699<\/td>\n<td>ISRIB (trans-isomer)<\/td>\n<\/tr>\n<tr>\n<td>A1910<\/td>\n<td>Bromodomain Inhibitor, (+)-JQ1<\/td>\n<\/tr>\n<tr>\n<td>B1293<\/td>\n<td>Y-27632<\/td>\n<\/tr>\n<tr>\n<td>A8167<\/td>\n<td>Rapamycin (Sirolimus)<\/td>\n<\/tr>\n<tr>\n<td>A7024<\/td>\n<td>HOAt<\/td>\n<\/tr>\n<tr>\n<td>A7025<\/td>\n<td>HOBt (anhydrous)<\/td>\n<\/tr>\n<tr>\n<td>A8331<\/td>\n<td>Bleomycin Sulfate<\/td>\n<\/tr>\n<tr>\n<td>A4333<\/td>\n<td>CPI-613<\/td>\n<\/tr>\n<tr>\n<td>K1070<\/td>\n<td>2X SYBR Green qPCR Master Mix<\/td>\n<\/tr>\n<tr>\n<td>A8005<\/td>\n<td>Sulfo-NHS-SS-Biotin<\/td>\n<\/tr>\n<tr>\n<td>B4653<\/td>\n<td>BV6<\/td>\n<\/tr>\n<tr>\n<td>B5965<\/td>\n<td>Tamoxifen<\/td>\n<\/tr>\n<tr>\n<td>A1901<\/td>\n<td>Q-VD-OPh hydrate<\/td>\n<\/tr>\n<tr>\n<td>A8950<\/td>\n<td>UM 171<\/td>\n<\/tr>\n<tr>\n<td>K1046<\/td>\n<td>RNase Inhibitor, Murine<\/td>\n<\/tr>\n<tr>\n<td>A3317<\/td>\n<td>Clozapine N-oxide (CNO)<\/td>\n<\/tr>\n<tr>\n<td>A2614<\/td>\n<td>Bortezomib (PS-341)<\/td>\n<\/tr>\n<tr>\n<td>A8003<\/td>\n<td>Sulfo-NHS-LC-Biotin<\/td>\n<\/tr>\n<tr>\n<td>A4154<\/td>\n<td>Olaparib (AZD2281, Ku-0059436)<\/td>\n<\/tr>\n<tr>\n<td>A8012<\/td>\n<td>Biotin-XX Tyramide Reagent<\/td>\n<\/tr>\n<tr>\n<td>K1101<\/td>\n<td>PreScission Protease (PSP)<\/td>\n<\/tr>\n<tr>\n<td>A8627<\/td>\n<td>Bafilomycin A1<\/td>\n<\/tr>\n<tr>\n<td>A8001<\/td>\n<td>Sulfo-NHS-Biotin<\/td>\n<\/tr>\n<tr>\n<td>A3017<\/td>\n<td>Dasatinib (BMS-354825)<\/td>\n<\/tr>\n<tr>\n<td>A2576<\/td>\n<td>E-64<\/td>\n<\/tr>\n<tr>\n<td>K1051<\/td>\n<td>Cy3 TSA Fluorescence System Kit<\/td>\n<\/tr>\n<tr>\n<td>K1034<\/td>\n<td>2X Taq PCR Master Mix (with dye)<\/td>\n<\/tr>\n<tr>\n<td>B7972<\/td>\n<td>Pseudo-UTP<\/td>\n<\/tr>\n<tr>\n<td>A8173<\/td>\n<td>Romidepsin (FK228, depsipeptide)<\/td>\n<\/tr>\n<tr>\n<td>A4219<\/td>\n<td>Birinapant (TL32711)<\/td>\n<\/tr>\n<tr>\n<td>A4371<\/td>\n<td>Ferrostatin-1 (Fer-1)<\/td>\n<\/tr>\n<tr>\n<td>A8200<\/td>\n<td>DAPT (GSI-IX)<\/td>\n<\/tr>\n<tr>\n<td>A8249<\/td>\n<td>SB 431542<\/td>\n<\/tr>\n<tr>\n<td>K1008<\/td>\n<td>Protease Inhibitor Cocktail (EDTA-Free, 200X in DMSO)<\/td>\n<\/tr>\n<tr>\n<td>A3133<\/td>\n<td>A 83-01<\/td>\n<\/tr>\n<tr>\n<td>A8192<\/td>\n<td>Staurosporine<\/td>\n<\/tr>\n<tr>\n<td>B1054<\/td>\n<td>Resiquimod (R-848)<\/td>\n<\/tr>\n<tr>\n<td>A3018<\/td>\n<td>Trametinib (GSK1120212)<\/td>\n<\/tr>\n<tr>\n<td>A8184<\/td>\n<td>AICAR<\/td>\n<\/tr>\n<tr>\n<td>K1025<\/td>\n<td>Direct Mouse Genotyping Kit<\/td>\n<\/tr>\n<tr>\n<td>A2606<\/td>\n<td>Epoxomicin<\/td>\n<\/tr>\n<tr>\n<td>A6006<\/td>\n<td>Hexa His tag peptide<\/td>\n<\/tr>\n<tr>\n<td>A4393<\/td>\n<td>Paclitaxel (Taxol)<\/td>\n<\/tr>\n<tr>\n<td>A8315<\/td>\n<td>NU7441 (KU-57788)<\/td>\n<\/tr>\n<tr>\n<td>A4213<\/td>\n<td>Necrostatin-1<\/td>\n<\/tr>\n<tr>\n<td>A8885<\/td>\n<td>Ro 3306<\/td>\n<\/tr>\n<tr>\n<td>L1021<\/td>\n<td>DiscoveryProbe\u2122 FDA-approved Drug Library<\/td>\n<\/tr>\n<tr>\n<td>B1464<\/td>\n<td>KPT-330<\/td>\n<\/tr>\n<tr>\n<td>A8815<\/td>\n<td>SM-164<\/td>\n<\/tr>\n<tr>\n<td>B4879<\/td>\n<td>Blasticidin S HCl<\/td>\n<\/tr>\n<tr>\n<td>A8793<\/td>\n<td>N3-kethoxal<\/td>\n<\/tr>\n<tr>\n<td>K1047<\/td>\n<td>HyperScribe\u2122 T7 High Yield RNA Synthesis Kit<\/td>\n<\/tr>\n<tr>\n<td>A6004<\/td>\n<td>Influenza Hemagglutinin (HA) Peptide<\/td>\n<\/tr>\n<tr>\n<td>B1036<\/td>\n<td>MLN4924<\/td>\n<\/tr>\n<tr>\n<td>A8178<\/td>\n<td>Panobinostat (LBH589)<\/td>\n<\/tr>\n<tr>\n<td>A3963<\/td>\n<td>A-769662<\/td>\n<\/tr>\n<tr>\n<td>A3847<\/td>\n<td>SU5416<\/td>\n<\/tr>\n<tr>\n<td>B3252<\/td>\n<td>Dorsomorphin (Compound C)<\/td>\n<\/tr>\n<tr>\n<td>B4758<\/td>\n<td>BAPTA-AM<\/td>\n<\/tr>\n<tr>\n<td>A2513<\/td>\n<td>Geneticin, G-418 Sulfate<\/td>\n<\/tr>\n<tr>\n<td>B6004<\/td>\n<td>PX-478 2HCl<\/td>\n<\/tr>\n<tr>\n<td>A8955<\/td>\n<td>Z-YVAD-FMK<\/td>\n<\/tr>\n<tr>\n<td>A8193<\/td>\n<td>ABT-737<\/td>\n<\/tr>\n<tr>\n<td>B2083<\/td>\n<td>Caspofungin Acetate<\/td>\n<\/tr>\n<tr>\n<td>A8002<\/td>\n<td>NHS-Biotin<\/td>\n<\/tr>\n<tr>\n<td>A8337<\/td>\n<td>CX-5461<\/td>\n<\/tr>\n<tr>\n<td>A8312<\/td>\n<td>Torin 1<\/td>\n<\/tr>\n<tr>\n<td>A2570<\/td>\n<td>Leupeptin, Microbial<\/td>\n<\/tr>\n<tr>\n<td>K2170<\/td>\n<td>Alanine Aminotransferase (ALT or SGPT) Activity Colorimetric\/Fluorometric Assay Kit<\/td>\n<\/tr>\n<tr>\n<td>A4381<\/td>\n<td>FK866 (APO866)<\/td>\n<\/tr>\n<tr>\n<td>B2143<\/td>\n<td>Tacrolimus (FK506)<\/td>\n<\/tr>\n<tr>\n<td>A2571<\/td>\n<td>Pepstatin A<\/td>\n<\/tr>\n<tr>\n<td>k1072<\/td>\n<td>First-Strand cDNA Synthesis Kit<\/td>\n<\/tr>\n<tr>\n<td>A3003<\/td>\n<td>MDV3100 (Enzalutamide)<\/td>\n<\/tr>\n<tr>\n<td>B5997<\/td>\n<td>Dyngo-4a<\/td>\n<\/tr>\n<tr>\n<td>A3742<\/td>\n<td>Pyridostatin<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<p><a href=\"http:\/\/www.apexbt.com\/\">APExBIO\u53f0\u7063\u4ee3\u7406\u5546<\/a><\/p>\n<p>APExBIO\u63d0\u4f9b\u512a\u8cea\u7684\u80dc\u80bd\u548c\u751f\u7269\u5206\u6790\u8a66\u5291\uff0c\u5ee3\u6cdb\u7522\u54c1\u7dda\u5982Protease\u3001Chromatin\/Epigenetics\u8868\u89c0\u907a\u50b3\u5b78\u3001MAPK Signal\u3001DNA Damege\/DNA repair\u3001\u7d30\u80de\u51cb\u4ea1\u3001\u816b\u7624\u751f\u7269\u5b78\u3001Stem cell\u7b49\u7814\u7a76\u9818\u57df\uff0c \u9084\u63d0\u4f9b\u5b9a\u5236\u7684\u670d\u52d9\uff0c\u5305\u62ec\u591a\u80bd\u5408\u6210\uff0c\u6297\u9ad4\u7684\u751f\u7522\u548c\u6aa2\u6e2c\u7684\u767c\u5c55\u3002\u7522\u54c1\u7ddaDNA\/RNA prep kit\u3001Drug Screening panel\u3001Bioactive peptides\u3001Growth factors\u3001Biotinylation Reagents\u3001tag peptides\u3001amino Acids\u3001Growth factors\u7b49\u3002APExBIO\u7522\u54c1\u8cea\u91cf\u90fd\u4f34\u96a8\u8457\u8b49\u66f8\u7684\u5206\u6790\uff0c\u9ad8\u6548\u6db2\u76f8\u8272\u8b5c\uff0c\u8cea\u8b5c\uff0c\u548cHMNR\u6578\u64da\u3002<\/p>\n<table width=\"1075\">\n<tbody>\n<tr>\n<td width=\"96\">A3477<\/td>\n<td width=\"375\">HOKU-81<\/td>\n<td width=\"158\">58020-43-2<\/td>\n<td width=\"79\">98.00%<\/td>\n<td width=\"367\">Bronchodilators,metabolite of tulobuterol<\/td>\n<\/tr>\n<tr>\n<td>A3478<\/td>\n<td>Hydroxyfasudil<\/td>\n<td>105628-72-6<\/td>\n<td>98.00%<\/td>\n<td>Rho-kinase inhibitor and vasodilator<\/td>\n<\/tr>\n<tr>\n<td>A3479<\/td>\n<td>Hydroxyfasudil hydrochloride<\/td>\n<td>155558-32-0<\/td>\n<td>98.71%<\/td>\n<td>Rho-kinase inhibitor and vasodilator<\/td>\n<\/tr>\n<tr>\n<td>A3481<\/td>\n<td>Ibutamoren Mesylate<\/td>\n<td>159752-10-0<\/td>\n<td>98.00%<\/td>\n<td>Growth hormone (GH) secretagogue<\/td>\n<\/tr>\n<tr>\n<td>A3482<\/td>\n<td>Icotinib Hydrochloride<\/td>\n<td>1204313-51-8<\/td>\n<td>98.00%<\/td>\n<td>EGFR inhibitor,potent and specific<\/td>\n<\/tr>\n<tr>\n<td>A3483<\/td>\n<td>IDO inhibitor 1<\/td>\n<td>1204669-37-3<\/td>\n<td>99.83%<\/td>\n<td>Indoleamine-2,3-dioxygenase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3484<\/td>\n<td>Iguratimod<\/td>\n<td>123663-49-0<\/td>\n<td>98.00%<\/td>\n<td>COX-2 inhibitor,inhibits IL-1,IL-6,IL-8 and tumour necrosis factor.<\/td>\n<\/tr>\n<tr>\n<td>A3485<\/td>\n<td>IKK-2 inhibitor VIII<\/td>\n<td>406209-26-5<\/td>\n<td>98.00%<\/td>\n<td>IKK-2 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3486<\/td>\n<td>IKK-3 Inhibitor<\/td>\n<td>862812-98-4<\/td>\n<td>98.00%<\/td>\n<td>IKK-3 Inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3487<\/td>\n<td>Imatinib hydrochloride<\/td>\n<td>862366-25-4<\/td>\n<td>98.00%<\/td>\n<td>V-Abl\/c-Kit\/PDGFR inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3492<\/td>\n<td>INCB 3284 dimesylate<\/td>\n<td>887401-93-6<\/td>\n<td>98.00%<\/td>\n<td>HCCR2 antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3493<\/td>\n<td>INCB024360 analogue<\/td>\n<td>914471-09-3<\/td>\n<td>99.81%<\/td>\n<td>potent and selective inhibitor of IDO1<\/td>\n<\/tr>\n<tr>\n<td>A3494<\/td>\n<td>INCB3344<\/td>\n<td>1262238-11-8<\/td>\n<td>98.01%<\/td>\n<td>CCR2 chemokine receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3495<\/td>\n<td>INCB8761(PF-4136309)<\/td>\n<td>1341224-83-6<\/td>\n<td>98.00%<\/td>\n<td>CCR2 Antagonist,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3496<\/td>\n<td>Indacaterol<\/td>\n<td>312753-06-3<\/td>\n<td>98.00%<\/td>\n<td>\u03b22-agonist<\/td>\n<\/tr>\n<tr>\n<td>A3498<\/td>\n<td>Inolitazone<\/td>\n<td>223132-37-4<\/td>\n<td>98.00%<\/td>\n<td>PPARgamma agonist<\/td>\n<\/tr>\n<tr>\n<td>A3499<\/td>\n<td>Inolitazone dihydrochloride<\/td>\n<td>223132-38-5<\/td>\n<td>98.00%<\/td>\n<td>PPAR\u03b3 agonist,high-affinity and novel<\/td>\n<\/tr>\n<tr>\n<td>A3500<\/td>\n<td>IRAK inhibitor 1<\/td>\n<td>1042224-63-4<\/td>\n<td>98.11%<\/td>\n<td>IRAK-4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3501<\/td>\n<td>IRAK inhibitor 2<\/td>\n<td>928333-30-6<\/td>\n<td>98.00%<\/td>\n<td>IRAK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3502<\/td>\n<td>IRAK inhibitor 3<\/td>\n<td>1012343-93-9<\/td>\n<td>98.00%<\/td>\n<td>IRAK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3503<\/td>\n<td>IRAK inhibitor 4<\/td>\n<td>1012104-68-5<\/td>\n<td>98.00%<\/td>\n<td>IRAK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3504<\/td>\n<td>IRAK inhibitor 6<\/td>\n<td>1042672-97-8<\/td>\n<td>99.90%<\/td>\n<td>IRAK-4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3505<\/td>\n<td>IRAK-1-4 Inhibitor I<\/td>\n<td>509093-47-4<\/td>\n<td>98.17%<\/td>\n<td>IRAK-1\/4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3506<\/td>\n<td>Isobavachalcone<\/td>\n<td>20784-50-3<\/td>\n<td>98.00%<\/td>\n<td>Diverse biological activity compound<\/td>\n<\/tr>\n<tr>\n<td>A3507<\/td>\n<td>Istaroxime<\/td>\n<td>203737-93-3<\/td>\n<td>98.00%<\/td>\n<td>Na+\/K+ ATPase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3508<\/td>\n<td>Istaroxime hydrochloride<\/td>\n<td>374559-48-5<\/td>\n<td>98.00%<\/td>\n<td>Inhibitor of Na+\/K+ ATPase<\/td>\n<\/tr>\n<tr>\n<td>A3510<\/td>\n<td>Ivacaftor benzenesulfonate<\/td>\n<td>1134822-09-5<\/td>\n<td>99.90%<\/td>\n<td>CFTR Potentiator<\/td>\n<\/tr>\n<tr>\n<td>A3511<\/td>\n<td>Ivacaftor hydrate<\/td>\n<td>1134822-07-3<\/td>\n<td>98.00%<\/td>\n<td>CFTR Potentiator<\/td>\n<\/tr>\n<tr>\n<td>A3512<\/td>\n<td>IWP-2<\/td>\n<td>686770-61-6<\/td>\n<td>98.00%<\/td>\n<td>Wnt production inhibitor,PORCN inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3513<\/td>\n<td>Ixabepilone<\/td>\n<td>219989-84-1<\/td>\n<td>98.00%<\/td>\n<td>Epothilone B analog;microtubule-stabilizing agent<\/td>\n<\/tr>\n<tr>\n<td>A3515<\/td>\n<td>JANEX-1<\/td>\n<td>202475-60-3<\/td>\n<td>99.27%<\/td>\n<td>JAK3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3516<\/td>\n<td>JC-1<\/td>\n<td>3520-43-2<\/td>\n<td>98.00%<\/td>\n<td>Probe for Mitochondrial Membrane Potential<\/td>\n<\/tr>\n<tr>\n<td>A3517<\/td>\n<td>JDTic<\/td>\n<td>361444-66-8<\/td>\n<td>98.00%<\/td>\n<td>Opioid antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3518<\/td>\n<td>JDTic 2HCl<\/td>\n<td>785835-79-2<\/td>\n<td>98.00%<\/td>\n<td>\u03ba-opioid receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3519<\/td>\n<td>JNK-IN-7<\/td>\n<td>1408064-71-0<\/td>\n<td>98.13%<\/td>\n<td>Selective JNK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3520<\/td>\n<td>JNK-IN-8<\/td>\n<td>1410880-22-6<\/td>\n<td>99.45%<\/td>\n<td>JNK inhibitor, selective and irreversible<\/td>\n<\/tr>\n<tr>\n<td>A3522<\/td>\n<td>Kaempferide<\/td>\n<td>491-54-3<\/td>\n<td>99.53%<\/td>\n<td>O-methylated flavonol<\/td>\n<\/tr>\n<tr>\n<td>A3524<\/td>\n<td>kb NB 142-70<\/td>\n<td>1233533-04-4<\/td>\n<td>98.21%<\/td>\n<td>Inhibitor of protein kinase D,selective<\/td>\n<\/tr>\n<tr>\n<td>A3525<\/td>\n<td>KB-R7943 mesylate<\/td>\n<td>182004-65-5<\/td>\n<td>98.75%<\/td>\n<td>Inhibitor of the reverse mode of the Na+\/Ca2+ exchanger<\/td>\n<\/tr>\n<tr>\n<td>A3526<\/td>\n<td>Ketone Ester<\/td>\n<td>1208313-97-6<\/td>\n<td>98.00%<\/td>\n<td>Delaies CNS-OT seizures in rats<\/td>\n<\/tr>\n<tr>\n<td>A3527<\/td>\n<td>Ki20227<\/td>\n<td>623142-96-1<\/td>\n<td>98.43%<\/td>\n<td>C-Fms tyrosine kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3528<\/td>\n<td>Kinetin<\/td>\n<td>525-79-1<\/td>\n<td>99.89%<\/td>\n<td>Plant growth hormones<\/td>\n<\/tr>\n<tr>\n<td>A3529<\/td>\n<td>KN-92<\/td>\n<td>176708-42-2<\/td>\n<td>99.55%<\/td>\n<td>CaMKII inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3530<\/td>\n<td>KN-92 hydrochloride<\/td>\n<td>1431698-47-3<\/td>\n<td>99.89%<\/td>\n<td>Inactive derivative of KN-93,control compound<\/td>\n<\/tr>\n<tr>\n<td>A3531<\/td>\n<td>KN-92 phosphate<\/td>\n<td>1135280-28-2<\/td>\n<td>99.35%<\/td>\n<td>CaMKII inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3532<\/td>\n<td>KN-93<\/td>\n<td>139298-40-1<\/td>\n<td>99.83%<\/td>\n<td>CaMKII inhibitor,selective and cometitive<\/td>\n<\/tr>\n<tr>\n<td>A3533<\/td>\n<td>Ko 143<\/td>\n<td>461054-93-3<\/td>\n<td>98.00%<\/td>\n<td>BCRP inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3534<\/td>\n<td>KU14R<\/td>\n<td>189224-48-4<\/td>\n<td>98.00%<\/td>\n<td>I(3)-R antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3535<\/td>\n<td>KX2-391 dihydrochloride<\/td>\n<td>1038395-65-1<\/td>\n<td>98.00%<\/td>\n<td>Src kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3536<\/td>\n<td>L-165041<\/td>\n<td>79558-09-1<\/td>\n<td>98.30%<\/td>\n<td>PPAR\u03b2\/\u03b4 agonist,cell permeable,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3538<\/td>\n<td>Laropiprant<\/td>\n<td>571170-77-9<\/td>\n<td>98.00%<\/td>\n<td>DP1 receptor antagonist,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3539<\/td>\n<td>Lck Inhibitor<\/td>\n<td>847950-09-8<\/td>\n<td>98.00%<\/td>\n<td>Lck inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3541<\/td>\n<td>LCL161<\/td>\n<td>1005342-46-0<\/td>\n<td>99.81%<\/td>\n<td>Antagonist of IAPs inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3542<\/td>\n<td>LCQ-908<\/td>\n<td>956136-95-1<\/td>\n<td>98.00%<\/td>\n<td>DGAT1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3543<\/td>\n<td>LDE225 Diphosphate<\/td>\n<td>1218778-77-8<\/td>\n<td>99.83%<\/td>\n<td>Smo antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3544<\/td>\n<td>LDK378 dihydrochloride<\/td>\n<td>1380575-43-8<\/td>\n<td>99.93%<\/td>\n<td>ALK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3545<\/td>\n<td>LDN193189 Hydrochloride<\/td>\n<td>1062368-62-0<\/td>\n<td>98.76%<\/td>\n<td>ALK inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3548<\/td>\n<td>Lersivirine<\/td>\n<td>473921-12-9<\/td>\n<td>98.00%<\/td>\n<td>NNRT inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3549<\/td>\n<td>Lesinurad<\/td>\n<td>878672-00-5<\/td>\n<td>99.77%<\/td>\n<td>URAT1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3550<\/td>\n<td>Letermovir<\/td>\n<td>917389-32-3<\/td>\n<td>99.52%<\/td>\n<td>Novel anti-CMV compound<\/td>\n<\/tr>\n<tr>\n<td>A3551<\/td>\n<td>Leuprolide Acetate<\/td>\n<td>74381-53-6<\/td>\n<td>99.74%<\/td>\n<td>Pituitary GnRH receptors agonist<\/td>\n<\/tr>\n<tr>\n<td>A3552<\/td>\n<td>Levomefolate calcium<\/td>\n<td>151533-22-1<\/td>\n<td>99.44%<\/td>\n<td>Artificial form of folate<\/td>\n<\/tr>\n<tr>\n<td>A3555<\/td>\n<td>Limonin<\/td>\n<td>1180-71-8<\/td>\n<td>99.76%<\/td>\n<td>Carcinogenesis inhibitor and HIV-1 replication inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3556<\/td>\n<td>LKB1 (AAK1 dual inhibitor)<\/td>\n<td>1093222-27-5<\/td>\n<td>99.04%<\/td>\n<td>Pim-1 kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3558<\/td>\n<td>LRRK2-IN-1<\/td>\n<td>1234480-84-2<\/td>\n<td>99.18%<\/td>\n<td>LRRK2 inhibitor,cell-permeable and ATP competitive<\/td>\n<\/tr>\n<tr>\n<td>A3561<\/td>\n<td>Lu AE58054 Hydrochloride<\/td>\n<td>467458-02-2<\/td>\n<td>99.32%<\/td>\n<td>5-HT(6)R antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3562<\/td>\n<td>Lucidin<\/td>\n<td>478-08-0<\/td>\n<td>98.00%<\/td>\n<td>Natural component of Rubia tinctorum L<\/td>\n<\/tr>\n<tr>\n<td>A3563<\/td>\n<td>LUF6000<\/td>\n<td>890087-21-5<\/td>\n<td>98.00%<\/td>\n<td>A3 AR modulator<\/td>\n<\/tr>\n<tr>\n<td>A3564<\/td>\n<td>Luliconazole<\/td>\n<td>187164-19-8<\/td>\n<td>99.20%<\/td>\n<td>Azole antifungal agent(interdigital tinea pedis)<\/td>\n<\/tr>\n<tr>\n<td>A3565<\/td>\n<td>LX-1031<\/td>\n<td>945976-76-1<\/td>\n<td>99.50%<\/td>\n<td>TPH inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3566<\/td>\n<td>LX1606<\/td>\n<td>1137608-69-5<\/td>\n<td>98.00%<\/td>\n<td>Tryptophan hydroxylase (TPH) inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3567<\/td>\n<td>LX-4211<\/td>\n<td>1018899-04-1<\/td>\n<td>99.67%<\/td>\n<td>SGLT1\/SGLT2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3568<\/td>\n<td>LY 303511<\/td>\n<td>154447-38-8<\/td>\n<td>98.00%<\/td>\n<td>MTOR inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3569<\/td>\n<td>LY 344864<\/td>\n<td>186544-26-3<\/td>\n<td>98.00%<\/td>\n<td>5-HT1F receptor agonist,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3570<\/td>\n<td>LY2090314<\/td>\n<td>603288-22-8<\/td>\n<td>99.78%<\/td>\n<td>Potent GSK-3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3571<\/td>\n<td>LY2183240<\/td>\n<td>874902-19-9<\/td>\n<td>98.00%<\/td>\n<td>Blocker of anandamide uptake,highly potent<\/td>\n<\/tr>\n<tr>\n<td>A3573<\/td>\n<td>LY2801653<\/td>\n<td>1206799-15-6<\/td>\n<td>99.47%<\/td>\n<td>MET inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3575<\/td>\n<td>LY2835219 free base<\/td>\n<td>1231929-97-7<\/td>\n<td>99.42%<\/td>\n<td>CDK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3576<\/td>\n<td>LY2874455<\/td>\n<td>1254473-64-7<\/td>\n<td>98.94%<\/td>\n<td>FGF\/FGFR Inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3577<\/td>\n<td>LY341495<\/td>\n<td>201943-63-7<\/td>\n<td>98.00%<\/td>\n<td>Metabotropic glutamate receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3583<\/td>\n<td>Matrine<\/td>\n<td>519-02-8<\/td>\n<td>98.87%<\/td>\n<td>Alkaloid found in Sophora plant<\/td>\n<\/tr>\n<tr>\n<td>A3584<\/td>\n<td>Maxacalcitol<\/td>\n<td>103909-75-7<\/td>\n<td>98.00%<\/td>\n<td>Non-calcemic vitamin D3 analog and VDR ligand.<\/td>\n<\/tr>\n<tr>\n<td>A3586<\/td>\n<td>MB05032<\/td>\n<td>261365-11-1<\/td>\n<td>98.00%<\/td>\n<td>GNG inhibitor,special and efficacious<\/td>\n<\/tr>\n<tr>\n<td>A3587<\/td>\n<td>MBX-2982<\/td>\n<td>1037792-44-1<\/td>\n<td>98.00%<\/td>\n<td>GPR119 agonist,selective and orally-available<\/td>\n<\/tr>\n<tr>\n<td>A3588<\/td>\n<td>MC 1046<\/td>\n<td>126860-83-1<\/td>\n<td>98.00%<\/td>\n<td>Vitamin D3 analog<\/td>\n<\/tr>\n<tr>\n<td>A3592<\/td>\n<td>Medetomidine<\/td>\n<td>86347-14-0<\/td>\n<td>98.00%<\/td>\n<td>\u03b12-adrenoceptor agonist<\/td>\n<\/tr>\n<tr>\n<td>A3593<\/td>\n<td>Mefloquine hydrochloride<\/td>\n<td>51773-92-3<\/td>\n<td>99.86%<\/td>\n<td>Quinoline methanol antimalarial agent,<\/td>\n<\/tr>\n<tr>\n<td>A3594<\/td>\n<td>MEK inhibitor<\/td>\n<td>334951-92-7<\/td>\n<td>98.00%<\/td>\n<td>Potent MEK inhibitor, Antitumor agent<\/td>\n<\/tr>\n<tr>\n<td>A3599<\/td>\n<td>Metoclopramide<\/td>\n<td>364-62-5<\/td>\n<td>99.94%<\/td>\n<td>Dopamine receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3600<\/td>\n<td>MF63<\/td>\n<td>892549-43-8<\/td>\n<td>98.00%<\/td>\n<td>MPGES-1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3601<\/td>\n<td>mGlu2 agonist<\/td>\n<td>1311385-32-6<\/td>\n<td>98.00%<\/td>\n<td>Anti-depressants,novel potent agent<\/td>\n<\/tr>\n<tr>\n<td>A3602<\/td>\n<td>MI-2<\/td>\n<td>1271738-62-5<\/td>\n<td>99.65%<\/td>\n<td>Menin-MLL Inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3603<\/td>\n<td>MI-3<\/td>\n<td>1271738-59-0<\/td>\n<td>98.00%<\/td>\n<td>Menin-MLL Inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3604<\/td>\n<td>Mibefradil<\/td>\n<td>116644-53-2<\/td>\n<td>98.07%<\/td>\n<td>Calcium channel blocker<\/td>\n<\/tr>\n<tr>\n<td>A3605<\/td>\n<td>Mibefradil dihydrochloride<\/td>\n<td>116666-63-8<\/td>\n<td>98.00%<\/td>\n<td>Ca2+ channel blocker ,antihypertensive<\/td>\n<\/tr>\n<tr>\n<td>A3606<\/td>\n<td>Micafungin sodium<\/td>\n<td>208538-73-2<\/td>\n<td>99.56%<\/td>\n<td>Inhibitor of \u03b2-(1,3)-D-glucan synthesis;fungicide<\/td>\n<\/tr>\n<tr>\n<td>A3608<\/td>\n<td>MK 0893<\/td>\n<td>870823-12-4<\/td>\n<td>98.58%<\/td>\n<td>Glucagon receptor\/IGF-1R antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3609<\/td>\n<td>MK-0591<\/td>\n<td>136668-42-3<\/td>\n<td>98.00%<\/td>\n<td>FLAP inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3611<\/td>\n<td>MK-0812<\/td>\n<td>624733-88-6<\/td>\n<td>98.00%<\/td>\n<td>antagonist of chemokine receptor CCR-2<\/td>\n<\/tr>\n<tr>\n<td>A3612<\/td>\n<td>MK-0974<\/td>\n<td>781649-09-0<\/td>\n<td>98.00%<\/td>\n<td>CGRP receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3613<\/td>\n<td>MK-2894<\/td>\n<td>1006036-87-8<\/td>\n<td>98.00%<\/td>\n<td>EP4 receptor inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3615<\/td>\n<td>MK-3207<\/td>\n<td>957118-49-9<\/td>\n<td>98.00%<\/td>\n<td>CGRP receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3617<\/td>\n<td>MK-4827<\/td>\n<td>1038915-60-4<\/td>\n<td>98.93%<\/td>\n<td>PARP-1\/-2 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3618<\/td>\n<td>MK-5172<\/td>\n<td>1350514-68-9<\/td>\n<td>99.79%<\/td>\n<td>HCV NS3\/4a protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3619<\/td>\n<td>MK-5172 hydrate<\/td>\n<td>1350462-55-3<\/td>\n<td>98.00%<\/td>\n<td>HCV NS3\/4a protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3620<\/td>\n<td>MK-5172 potassium salt<\/td>\n<td>1206524-86-8<\/td>\n<td>98.00%<\/td>\n<td>HCV NS3\/4a protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3621<\/td>\n<td>MK-5172 sodium salt<\/td>\n<td>1425038-27-2<\/td>\n<td>98.00%<\/td>\n<td>HCV NS3\/4a protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3623<\/td>\n<td>MK-6892<\/td>\n<td>917910-45-3<\/td>\n<td>99.65%<\/td>\n<td>Highly potential GPR109A agonist<\/td>\n<\/tr>\n<tr>\n<td>A3624<\/td>\n<td>MK-8033<\/td>\n<td>1001917-37-8<\/td>\n<td>98.00%<\/td>\n<td>C-MET inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3626<\/td>\n<td>ML-7 hydrochloride<\/td>\n<td>110448-33-4<\/td>\n<td>98.43%<\/td>\n<td>Myosin light chain kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3627<\/td>\n<td>MLN 2480<\/td>\n<td>1096708-71-2<\/td>\n<td>98.99%<\/td>\n<td>Pan-Raf kinase inhibitor,investigational<\/td>\n<\/tr>\n<tr>\n<td>A3628<\/td>\n<td>MLN120B<\/td>\n<td>783348-36-7<\/td>\n<td>99.82%<\/td>\n<td>I\u03baB Kinase \u03b2 Inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3629<\/td>\n<td>MLN4924 HCl salt<\/td>\n<td>1160295-21-5<\/td>\n<td>98.00%<\/td>\n<td>NAE inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3630<\/td>\n<td>MMAD<\/td>\n<td>203849-91-6<\/td>\n<td>98.00%<\/td>\n<td>Tubulin inhibitor,highly potent<\/td>\n<\/tr>\n<tr>\n<td>A3631<\/td>\n<td>Monomethyl auristatin E<\/td>\n<td>474645-27-7<\/td>\n<td>98.34%<\/td>\n<td>Antimitotic agent<\/td>\n<\/tr>\n<tr>\n<td>A3632<\/td>\n<td>Motesanib<\/td>\n<td>453562-69-1<\/td>\n<td>98.00%<\/td>\n<td>Inhibitor of Flk-1\/Flt-4\/PDGFR-\/c-Kit<\/td>\n<\/tr>\n<tr>\n<td>A3633<\/td>\n<td>MPEP Hydrochloride<\/td>\n<td>219911-35-0<\/td>\n<td>98.00%<\/td>\n<td>MGlu5 receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3634<\/td>\n<td>MPTP hydrochloride<\/td>\n<td>23007-85-4<\/td>\n<td>99.79%<\/td>\n<td>Dopaminergic neurotoxin,induced reduction in the DOPAC HVA\/dopamine (DA) ratio<\/td>\n<\/tr>\n<tr>\n<td>A3636<\/td>\n<td>MTEP hydrochloride<\/td>\n<td>1186195-60-7<\/td>\n<td>98.00%<\/td>\n<td>MGlu5 antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3637<\/td>\n<td>GDC-mTOR inhibitor<\/td>\n<td>1207358-59-5<\/td>\n<td>98.00%<\/td>\n<td>MTOR inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3641<\/td>\n<td>Naphthoquine phosphate<\/td>\n<td>173531-58-3<\/td>\n<td>98.00%<\/td>\n<td>Antimalarial drug<\/td>\n<\/tr>\n<tr>\n<td>A3642<\/td>\n<td>Narciclasine<\/td>\n<td>29477-83-6<\/td>\n<td>98.00%<\/td>\n<td>Modulates the Rho\/ROCK\/LIM kinase\/cofilin pathway<\/td>\n<\/tr>\n<tr>\n<td>A3643<\/td>\n<td>Narlaprevir<\/td>\n<td>865466-24-6<\/td>\n<td>98.00%<\/td>\n<td>HCV NS3 protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3645<\/td>\n<td>NB-598<\/td>\n<td>131060-14-5<\/td>\n<td>99.35%<\/td>\n<td>SE inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3646<\/td>\n<td>NB-598 hydrochloride<\/td>\n<td>136719-25-0<\/td>\n<td>98.00%<\/td>\n<td>SE inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3647<\/td>\n<td>NB-598 Maleate<\/td>\n<td>155294-62-5<\/td>\n<td>98.97%<\/td>\n<td>Squalene epoxidase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3649<\/td>\n<td>NBD-556<\/td>\n<td>333353-44-9<\/td>\n<td>98.00%<\/td>\n<td>HIV-1 entry inhibitor,CD4 mimetic,block gp120-CD4 interaction<\/td>\n<\/tr>\n<tr>\n<td>A3652<\/td>\n<td>Necrostatin 2<\/td>\n<td>852391-19-6<\/td>\n<td>98.00%<\/td>\n<td>In vitro necroptosis inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3653<\/td>\n<td>Nelfinavir Mesylate<\/td>\n<td>159989-65-8<\/td>\n<td>98.04%<\/td>\n<td>HIV protease inhibitor,antiretroviral drug for HIV treatment<\/td>\n<\/tr>\n<tr>\n<td>A3655<\/td>\n<td>Nesbuvir<\/td>\n<td>691852-58-1<\/td>\n<td>99.79%<\/td>\n<td>NS5B polymerase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3658<\/td>\n<td>NG25<\/td>\n<td>1315355-93-1<\/td>\n<td>98.00%<\/td>\n<td>TAK1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3659<\/td>\n<td>Nifuratel<\/td>\n<td>4936-47-4<\/td>\n<td>98.00%<\/td>\n<td>Antibacterial, antifungal, and antiprotozoal compound<\/td>\n<\/tr>\n<tr>\n<td>A3660<\/td>\n<td>Nilotinib monohydrochloride monohydrate<\/td>\n<td>923288-90-8<\/td>\n<td>99.89%<\/td>\n<td>Bcr-Abl inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3662<\/td>\n<td>NNC 55-0396<\/td>\n<td>357400-13-6<\/td>\n<td>98.00%<\/td>\n<td>T-type calcium channel blocker<\/td>\n<\/tr>\n<tr>\n<td>A3663<\/td>\n<td>Noopept<\/td>\n<td>157115-85-0<\/td>\n<td>98.00%<\/td>\n<td>Nootropic and neuroprotective agent<\/td>\n<\/tr>\n<tr>\n<td>A3664<\/td>\n<td>Nordihydroguaiaretic acid<\/td>\n<td>500-38-9<\/td>\n<td>99.83%<\/td>\n<td>Anti-tumor agent;lipoxygenase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3665<\/td>\n<td>Nortadalafil<\/td>\n<td>171596-36-4<\/td>\n<td>98.00%<\/td>\n<td>PDE5 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3666<\/td>\n<td>NP118809<\/td>\n<td>41332-24-5<\/td>\n<td>98.00%<\/td>\n<td>N-type calcium channel blocker<\/td>\n<\/tr>\n<tr>\n<td>A3667<\/td>\n<td>NPS-2143 hydrochloride<\/td>\n<td>324523-20-8<\/td>\n<td>99.89%<\/td>\n<td>Calcium ion-sensing receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3668<\/td>\n<td>NS309<\/td>\n<td>18711-16-5<\/td>\n<td>98.00%<\/td>\n<td>Calcium-Activated Potassium Channel activator<\/td>\n<\/tr>\n<tr>\n<td>A3670<\/td>\n<td>Nucleozin<\/td>\n<td>341001-38-5<\/td>\n<td>99.55%<\/td>\n<td>Targets influenza A nucleoprotein (NP),cell-permeable isoxazolylpiperazine compound<\/td>\n<\/tr>\n<tr>\n<td>A3671<\/td>\n<td>Nutlin-3a chiral<\/td>\n<td>675576-98-4<\/td>\n<td>98.39%<\/td>\n<td>MDM2 inhibitor, antiproliferative and antiproapoptotic<\/td>\n<\/tr>\n<tr>\n<td>A3672<\/td>\n<td>NVP-BAG956<\/td>\n<td>853910-02-8<\/td>\n<td>98.00%<\/td>\n<td>PI3K and PDK1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3673<\/td>\n<td>NVP-BGJ398 phosphate<\/td>\n<td>1310746-10-1<\/td>\n<td>99.78%<\/td>\n<td>FGFR inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3674<\/td>\n<td>NVP-BKM120 Hydrochloride<\/td>\n<td>1312445-63-8<\/td>\n<td>98.02%<\/td>\n<td>PI3K inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3675<\/td>\n<td>NVP-BSK805<\/td>\n<td>1092499-93-8<\/td>\n<td>98.00%<\/td>\n<td>ATP-competitive JAK2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3676<\/td>\n<td>NVP-LCQ195<\/td>\n<td>902156-99-4<\/td>\n<td>97.50%<\/td>\n<td>CDK1\/CDK2\/CDK5 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3680<\/td>\n<td>Olcegepant<\/td>\n<td>204697-65-4<\/td>\n<td>97.46%<\/td>\n<td>Non-peptide receptor of CGRP,first potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3681<\/td>\n<td>Olmesartan<\/td>\n<td>144689-24-7<\/td>\n<td>99.20%<\/td>\n<td>Angiotensin II receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3683<\/td>\n<td>Olprinone Hydrochloride<\/td>\n<td>119615-63-3<\/td>\n<td>99.74%<\/td>\n<td>Phosphodiesterase 3 (PDE3) inhibitor, selective<\/td>\n<\/tr>\n<tr>\n<td>A3684<\/td>\n<td>ONO-AE3-208<\/td>\n<td>402473-54-5<\/td>\n<td>97.73%<\/td>\n<td>EP4 receptor antagonist,high affinity and selective<\/td>\n<\/tr>\n<tr>\n<td>A3686<\/td>\n<td>Orteronel<\/td>\n<td>566939-85-3<\/td>\n<td>98.00%<\/td>\n<td>For castration-resistant prostate cancer, clinical candidate<\/td>\n<\/tr>\n<tr>\n<td>A3688<\/td>\n<td>Oseltamivir<\/td>\n<td>196618-13-0<\/td>\n<td>96.83%<\/td>\n<td>inhibitor of influenza neuraminidase<\/td>\n<\/tr>\n<tr>\n<td>A3689<\/td>\n<td>Oseltamivir acid<\/td>\n<td>187227-45-8<\/td>\n<td>99.08%<\/td>\n<td>Influenza neuraminidase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3690<\/td>\n<td>Otamixaban<\/td>\n<td>193153-04-7<\/td>\n<td>98.00%<\/td>\n<td>Direct factor Xa inhibitors,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3691<\/td>\n<td>Otenabant<\/td>\n<td>686344-29-6<\/td>\n<td>98.00%<\/td>\n<td>CB1 receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3692<\/td>\n<td>OTX-015<\/td>\n<td>202590-98-5<\/td>\n<td>99.57%<\/td>\n<td>BRD inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3695<\/td>\n<td>Pafuramidine<\/td>\n<td>186953-56-0<\/td>\n<td>98.00%<\/td>\n<td>Prodrug of furamidine<\/td>\n<\/tr>\n<tr>\n<td>A3696<\/td>\n<td>Palifosfamide<\/td>\n<td>31645-39-3<\/td>\n<td>98.00%<\/td>\n<td>Active metabolite of ifosfamide (IFOS)<\/td>\n<\/tr>\n<tr>\n<td>A3697<\/td>\n<td>Palonosetron<\/td>\n<td>135729-61-2<\/td>\n<td>98.00%<\/td>\n<td>5-HT3 antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3700<\/td>\n<td>Paradol<\/td>\n<td>27113-22-0<\/td>\n<td>98.00%<\/td>\n<td>Active flavor constituent of the seeds of Guinea pepper<\/td>\n<\/tr>\n<tr>\n<td>A3702<\/td>\n<td>Paricalcitol<\/td>\n<td>131918-61-1<\/td>\n<td>98.00%<\/td>\n<td>Analog of VD2 active form<\/td>\n<\/tr>\n<tr>\n<td>A3704<\/td>\n<td>PD 123319 ditrifluoroacetate<\/td>\n<td>136676-91-0<\/td>\n<td>99.14%<\/td>\n<td>Angiotensin AT2 receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3706<\/td>\n<td>PDK1 inhibitor<\/td>\n<td>1001409-50-2<\/td>\n<td>98.00%<\/td>\n<td>PDK1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3707<\/td>\n<td>Pemetrexed disodium hemipenta hydrate<\/td>\n<td>357166-30-4<\/td>\n<td>99.94%<\/td>\n<td>Antifolate and antimetabolite agent<\/td>\n<\/tr>\n<tr>\n<td>A3708<\/td>\n<td>Pentostatin<\/td>\n<td>53910-25-1<\/td>\n<td>99.05%<\/td>\n<td>Irreversible adenosine deaminase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3709<\/td>\n<td>Peramivir<\/td>\n<td>330600-85-6<\/td>\n<td>99.01%<\/td>\n<td>Aeuraminidase inhibitor;antiviral drug<\/td>\n<\/tr>\n<tr>\n<td>A3711<\/td>\n<td>PF-03084014<\/td>\n<td>865773-15-5<\/td>\n<td>98.52%<\/td>\n<td>\u03b3-secretase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3712<\/td>\n<td>PF-04217903 methanesulfonate<\/td>\n<td>956906-93-7<\/td>\n<td>98.00%<\/td>\n<td>C-Met inhibitor,selective and ATP-competitive<\/td>\n<\/tr>\n<tr>\n<td>A3715<\/td>\n<td>PF-04971729<\/td>\n<td>1210344-57-2<\/td>\n<td>98.00%<\/td>\n<td>SGLT inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3716<\/td>\n<td>PF-3758309<\/td>\n<td>898044-15-0<\/td>\n<td>98.39%<\/td>\n<td>PAK4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3717<\/td>\n<td>PF-543<\/td>\n<td>1415562-82-1<\/td>\n<td>99.32%<\/td>\n<td>SphK1 inhibitor,cell-permeate,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3718<\/td>\n<td>PF-543 Citrate<\/td>\n<td>1415562-83-2<\/td>\n<td>98.95%<\/td>\n<td>SphK1 inhibitor,potent and cell-permeate<\/td>\n<\/tr>\n<tr>\n<td>A3719<\/td>\n<td>PF-670462<\/td>\n<td>950912-80-8<\/td>\n<td>99.66%<\/td>\n<td>CK1 \u03b5\/\u03b4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3720<\/td>\n<td>PF-8380<\/td>\n<td>1144035-53-9<\/td>\n<td>98.23%<\/td>\n<td>Autotaxin inhibitor,potent and specific<\/td>\n<\/tr>\n<tr>\n<td>A3721<\/td>\n<td>PHA-767491<\/td>\n<td>845714-00-3<\/td>\n<td>99.03%<\/td>\n<td>Cdc7\/cdk9 inhibitor, potent, ATP-competitive<\/td>\n<\/tr>\n<tr>\n<td>A3722<\/td>\n<td>Phenylpiracetam<\/td>\n<td>77472-70-9<\/td>\n<td>99.21%<\/td>\n<td>Nootropic derivative of piracetam<\/td>\n<\/tr>\n<tr>\n<td>A3723<\/td>\n<td>Phloretin<\/td>\n<td>60-82-2<\/td>\n<td>99.12%<\/td>\n<td>A dihydrochalcone found in apple<\/td>\n<\/tr>\n<tr>\n<td>A3724<\/td>\n<td>PI-103 Hydrochloride<\/td>\n<td>371935-79-4<\/td>\n<td>98.00%<\/td>\n<td>DNA-PK\/PI 3-kinase\/mTOR inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3727<\/td>\n<td>Pitolisant hydrochloride<\/td>\n<td>903576-44-3<\/td>\n<td>99.71%<\/td>\n<td>Nonimidazole inverse agonist<\/td>\n<\/tr>\n<tr>\n<td>A3729<\/td>\n<td>PJ34<\/td>\n<td>344458-19-1<\/td>\n<td>95.69%<\/td>\n<td>PARP-l inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3730<\/td>\n<td>PND-1186<\/td>\n<td>1061353-68-1<\/td>\n<td>99.75%<\/td>\n<td>Potent FAK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3732<\/td>\n<td>Poloxin<\/td>\n<td>321688-88-4<\/td>\n<td>98.00%<\/td>\n<td>PLK1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3733<\/td>\n<td>Pramipexole dihydrochloride<\/td>\n<td>104632-25-9<\/td>\n<td>98.94%<\/td>\n<td>Dopamine receptor agonist<\/td>\n<\/tr>\n<tr>\n<td>A3735<\/td>\n<td>Preladenant<\/td>\n<td>377727-87-2<\/td>\n<td>98.00%<\/td>\n<td>Adenosine A2A receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3736<\/td>\n<td>PRT062607 Hydrochloride<\/td>\n<td>1370261-97-4<\/td>\n<td>98.63%<\/td>\n<td>SYK inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3738<\/td>\n<td>PSI-7977<\/td>\n<td>1190307-88-0<\/td>\n<td>99.81%<\/td>\n<td>Antiviral agents for chronic HCV infection<\/td>\n<\/tr>\n<tr>\n<td>A3740<\/td>\n<td>Puromycin aminonucleoside<\/td>\n<td>58-60-6<\/td>\n<td>98.19%<\/td>\n<td>Aminonucleoside portion of the antibiotic puromycin<\/td>\n<\/tr>\n<tr>\n<td>A3741<\/td>\n<td>Pyridone 6<\/td>\n<td>457081-03-7<\/td>\n<td>99.60%<\/td>\n<td>Pan-JAK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3742<\/td>\n<td>Pyridostatin<\/td>\n<td>1085412-37-8<\/td>\n<td>98.02%<\/td>\n<td>Drug used for promoting growth arrest<\/td>\n<\/tr>\n<tr>\n<td>A3744<\/td>\n<td>Quetiapine<\/td>\n<td>111974-69-7<\/td>\n<td>98.00%<\/td>\n<td>Dopamine receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3746<\/td>\n<td>R1530<\/td>\n<td>882531-87-5<\/td>\n<td>98.00%<\/td>\n<td>Antiangiogenesis,mitosis-angiogenesis inhibitor (MAI)<\/td>\n<\/tr>\n<tr>\n<td>A3747<\/td>\n<td>R-7128<\/td>\n<td>940908-79-2<\/td>\n<td>98.00%<\/td>\n<td>NS5B inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3749<\/td>\n<td>Radezolid<\/td>\n<td>869884-78-6<\/td>\n<td>99.32%<\/td>\n<td>Novel oxazolidinone antibiotic agent<\/td>\n<\/tr>\n<tr>\n<td>A3750<\/td>\n<td>Regorafenib hydrochloride<\/td>\n<td>835621-07-3<\/td>\n<td>98.57%<\/td>\n<td>Tyrosine kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3752<\/td>\n<td>Reparixin<\/td>\n<td>266359-83-5<\/td>\n<td>98.11%<\/td>\n<td>Inhibitor of CXCL8 receptor and CXCR1\/CXCR2 activation<\/td>\n<\/tr>\n<tr>\n<td>A3753<\/td>\n<td>Reparixin L-lysine salt<\/td>\n<td>266359-93-7<\/td>\n<td>97.82%<\/td>\n<td>CXCR1\/CXCR2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3754<\/td>\n<td>RepSox<\/td>\n<td>446859-33-2<\/td>\n<td>99.83%<\/td>\n<td>ALK5 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3755<\/td>\n<td>Resminostat hydrochloride<\/td>\n<td>1187075-34-8<\/td>\n<td>98.00%<\/td>\n<td>HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3756<\/td>\n<td>Retaspimycin<\/td>\n<td>857402-23-4<\/td>\n<td>98.00%<\/td>\n<td>HSP90 inhibitor,antiproliferative and antineoplastic<\/td>\n<\/tr>\n<tr>\n<td>A3758<\/td>\n<td>Retigabine dihydrochloride<\/td>\n<td>150812-13-8<\/td>\n<td>99.27%<\/td>\n<td>Antiepileptic compound<\/td>\n<\/tr>\n<tr>\n<td>A3759<\/td>\n<td>Retinyl glucoside<\/td>\n<td>136778-12-6<\/td>\n<td>98.00%<\/td>\n<td>Metabolites of vitamin A<\/td>\n<\/tr>\n<tr>\n<td>A3760<\/td>\n<td>Reversine<\/td>\n<td>656820-32-5<\/td>\n<td>99.09%<\/td>\n<td>A3 adenosine receptor antagonist,ARK-1\/-2\/-3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3761<\/td>\n<td>RG2833<\/td>\n<td>1215493-56-3<\/td>\n<td>98.06%<\/td>\n<td>Brain-penetrant HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3762<\/td>\n<td>RG7112<\/td>\n<td>939981-39-2<\/td>\n<td>98.58%<\/td>\n<td>MDM2 inhibitor, first clinical<\/td>\n<\/tr>\n<tr>\n<td>A3763<\/td>\n<td>RG7388<\/td>\n<td>1229705-06-9<\/td>\n<td>99.82%<\/td>\n<td>MDM2 antagonist, oral, selective<\/td>\n<\/tr>\n<tr>\n<td>A3764<\/td>\n<td>RI-1<\/td>\n<td>415713-60-9<\/td>\n<td>99.54%<\/td>\n<td>RAD51 inhibitor,cell-permeable<\/td>\n<\/tr>\n<tr>\n<td>A3765<\/td>\n<td>Rilpivirine<\/td>\n<td>500287-72-9<\/td>\n<td>99.64%<\/td>\n<td>Inhibitor of next-generation nonnucleoside reverse transcriptase<\/td>\n<\/tr>\n<tr>\n<td>A3766<\/td>\n<td>Rimonabant hydrochloride<\/td>\n<td>158681-13-1<\/td>\n<td>98.01%<\/td>\n<td>CB1 receptor inverse agonist<\/td>\n<\/tr>\n<tr>\n<td>A3767<\/td>\n<td>Riociguat<\/td>\n<td>625115-55-1<\/td>\n<td>99.77%<\/td>\n<td>Soluble guanylate cyclase (sGC) stimulator<\/td>\n<\/tr>\n<tr>\n<td>A3768<\/td>\n<td>Rivastigmine<\/td>\n<td>123441-03-2<\/td>\n<td>99.68%<\/td>\n<td>Cholinesterase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3770<\/td>\n<td>RJR-2403 oxalate<\/td>\n<td>220662-95-3<\/td>\n<td>98.00%<\/td>\n<td>Nicotinic receptor agonist<\/td>\n<\/tr>\n<tr>\n<td>A3771<\/td>\n<td>RKI-1447<\/td>\n<td>1342278-01-6<\/td>\n<td>99.52%<\/td>\n<td>Potent ROCK1\/ROCK2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3776<\/td>\n<td>Rotigotine<\/td>\n<td>99755-59-6<\/td>\n<td>98.00%<\/td>\n<td>Agonist of dopamine D2\/D3 receptor<\/td>\n<\/tr>\n<tr>\n<td>A3777<\/td>\n<td>Rotigotine hydrochloride<\/td>\n<td>125572-93-2<\/td>\n<td>98.00%<\/td>\n<td>Agonist of dopamine D2\/D3 receptor<\/td>\n<\/tr>\n<tr>\n<td>A3778<\/td>\n<td>RS 127445<\/td>\n<td>199864-87-4<\/td>\n<td>98.01%<\/td>\n<td>5-HT2B receptor antagonist,high affinity<\/td>\n<\/tr>\n<tr>\n<td>A3780<\/td>\n<td>RU 58841<\/td>\n<td>154992-24-2<\/td>\n<td>98.40%<\/td>\n<td>Androgen receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3781<\/td>\n<td>Ruxolitinib phosphate<\/td>\n<td>1092939-17-7<\/td>\n<td>98.75%<\/td>\n<td>JAK1\/JAK2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3783<\/td>\n<td>S0859<\/td>\n<td>1019331-10-2<\/td>\n<td>98.00%<\/td>\n<td>NBC inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3784<\/td>\n<td>Safinamide<\/td>\n<td>133865-89-1<\/td>\n<td>99.64%<\/td>\n<td>MAO-B inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3787<\/td>\n<td>Salirasib<\/td>\n<td>162520-00-5<\/td>\n<td>99.28%<\/td>\n<td>Inhibitor of active Ras protein<\/td>\n<\/tr>\n<tr>\n<td>A3789<\/td>\n<td>Salmeterol xinafoate<\/td>\n<td>94749-08-3<\/td>\n<td>98.11%<\/td>\n<td>\u03b22-adrenergic receptor agonist<\/td>\n<\/tr>\n<tr>\n<td>A3790<\/td>\n<td>Saquinavir<\/td>\n<td>127779-20-8<\/td>\n<td>98.00%<\/td>\n<td>HIV Protease Inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3791<\/td>\n<td>Saquinavir mesylate<\/td>\n<td>149845-06-7<\/td>\n<td>99.75%<\/td>\n<td>HIV Protease Inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3792<\/td>\n<td>SB 239063<\/td>\n<td>193551-21-2<\/td>\n<td>98.63%<\/td>\n<td>P38 MAP kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3794<\/td>\n<td>SB1317<\/td>\n<td>937270-47-8<\/td>\n<td>98.02%<\/td>\n<td>CDK,JAK and FLT inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3795<\/td>\n<td>SB-222200<\/td>\n<td>174635-69-9<\/td>\n<td>98.86%<\/td>\n<td>Human NK-3 receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3798<\/td>\n<td>SB-408124 Hydrochloride<\/td>\n<td>1431697-90-3<\/td>\n<td>98.00%<\/td>\n<td>OX1 receptor antagonist,selective and non-peptide<\/td>\n<\/tr>\n<tr>\n<td>A3800<\/td>\n<td>SB-674042<\/td>\n<td>483313-22-0<\/td>\n<td>98.00%<\/td>\n<td>OX1 selective antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3802<\/td>\n<td>SCH 527123<\/td>\n<td>473727-83-2<\/td>\n<td>99.40%<\/td>\n<td>CXCR1 and CXCR2 receptors antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3804<\/td>\n<td>SCH-1473759<\/td>\n<td>1094069-99-4<\/td>\n<td>98.00%<\/td>\n<td>Aurora A\/B inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3805<\/td>\n<td>SCH772984<\/td>\n<td>942183-80-4<\/td>\n<td>98.06%<\/td>\n<td>ERK1 and ERK2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3806<\/td>\n<td>SCH900776 S-isomer<\/td>\n<td>891494-64-7<\/td>\n<td>99.18%<\/td>\n<td>Checkpoint kinase(Chk)inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3808<\/td>\n<td>SD-208<\/td>\n<td>627536-09-8<\/td>\n<td>99.11%<\/td>\n<td>TGF-\u03b2R I kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3809<\/td>\n<td>SDZ 220-581<\/td>\n<td>174575-17-8<\/td>\n<td>98.00%<\/td>\n<td>NMDA glutamate receptor subtype antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3811<\/td>\n<td>SEA0400<\/td>\n<td>223104-29-8<\/td>\n<td>99.20%<\/td>\n<td>Specific inhibitor of Na+\/Ca2+ exchange<\/td>\n<\/tr>\n<tr>\n<td>A3814<\/td>\n<td>Seocalcitol<\/td>\n<td>134404-52-7<\/td>\n<td>98.00%<\/td>\n<td>Vitamin D receptor agonist<\/td>\n<\/tr>\n<tr>\n<td>A3815<\/td>\n<td>Setiptiline<\/td>\n<td>57262-94-9<\/td>\n<td>98.00%<\/td>\n<td>Serotonin receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3816<\/td>\n<td>Setiptiline maleate<\/td>\n<td>85650-57-3<\/td>\n<td>98.00%<\/td>\n<td>Serotonin receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3818<\/td>\n<td>Silvestrol<\/td>\n<td>697235-38-4<\/td>\n<td>98.00%<\/td>\n<td>Antineoplastic<\/td>\n<\/tr>\n<tr>\n<td>A3820<\/td>\n<td>Simeprevir<\/td>\n<td>923604-59-5<\/td>\n<td>99.42%<\/td>\n<td>Inhibitor of HCV NS3\/4A protease<\/td>\n<\/tr>\n<tr>\n<td>A3821<\/td>\n<td>SRT2104 (GSK2245840)<\/td>\n<td>1093403-33-8<\/td>\n<td>98.50%<\/td>\n<td>SIRT1 activator,selective<\/td>\n<\/tr>\n<tr>\n<td>A3823<\/td>\n<td>SJB2-043<\/td>\n<td>63388-44-3<\/td>\n<td>99.78%<\/td>\n<td>USP1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3824<\/td>\n<td>Skepinone-L<\/td>\n<td>1221485-83-1<\/td>\n<td>99.88%<\/td>\n<td>P38-MAPK inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3825<\/td>\n<td>SLx-2119<\/td>\n<td>911417-87-3<\/td>\n<td>98.80%<\/td>\n<td>Selective ROCK2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3826<\/td>\n<td>SMIP004<\/td>\n<td>143360-00-3<\/td>\n<td>98.17%<\/td>\n<td>Apoptosis inducer<\/td>\n<\/tr>\n<tr>\n<td>A3828<\/td>\n<td>Sobetirome<\/td>\n<td>211110-63-3<\/td>\n<td>99.01%<\/td>\n<td>Agonist of tyroid hormone receptor<\/td>\n<\/tr>\n<tr>\n<td>A3829<\/td>\n<td>sodium 4-pentynoate<\/td>\n<td>101917-30-0<\/td>\n<td>98.00%<\/td>\n<td>chemical reporter for the profiling of acetylated proteins<\/td>\n<\/tr>\n<tr>\n<td>A3832<\/td>\n<td>Solasodine<\/td>\n<td>126-17-0<\/td>\n<td>98.00%<\/td>\n<td>Neuroprotective antioxidant glycoalkaloid<\/td>\n<\/tr>\n<tr>\n<td>A3834<\/td>\n<td>SQ109<\/td>\n<td>502487-67-4<\/td>\n<td>98.00%<\/td>\n<td>Antibiotic for treatment of pulmonary TB<\/td>\n<\/tr>\n<tr>\n<td>A3835<\/td>\n<td>SR1078<\/td>\n<td>1246525-60-9<\/td>\n<td>98.65%<\/td>\n<td>Orphan receptor agonist<\/td>\n<\/tr>\n<tr>\n<td>A3836<\/td>\n<td>SR3335<\/td>\n<td>293753-05-6<\/td>\n<td>99.52%<\/td>\n<td>ROR\u03b1 agonist,partial inverse and selective<\/td>\n<\/tr>\n<tr>\n<td>A3837<\/td>\n<td>DL-\u03b1-Hydroxyglutaric acid disodium salt<\/td>\n<td>40951-21-1<\/td>\n<td>98.00%<\/td>\n<td>alpha hydroxy acid<\/td>\n<\/tr>\n<tr>\n<td>A3838<\/td>\n<td>SRT3109<\/td>\n<td>1204707-71-0<\/td>\n<td>98.00%<\/td>\n<td>CXCR2 ligand<\/td>\n<\/tr>\n<tr>\n<td>A3839<\/td>\n<td>SRT3190<\/td>\n<td>1204707-73-2<\/td>\n<td>99.56%<\/td>\n<td>CXCR2 ligand,SIRT1 activator<\/td>\n<\/tr>\n<tr>\n<td>A3840<\/td>\n<td>ST 2825<\/td>\n<td>894787-30-5<\/td>\n<td>98.00%<\/td>\n<td>Inhibitor of MyD88 dimerization<\/td>\n<\/tr>\n<tr>\n<td>A3843<\/td>\n<td>SU 5402<\/td>\n<td>215543-92-3<\/td>\n<td>98.48%<\/td>\n<td>VEGFR2\/FGFR\/PDGFR\/EGFR inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3844<\/td>\n<td>SU14813<\/td>\n<td>627908-92-3<\/td>\n<td>98.00%<\/td>\n<td>Tyrosine kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3846<\/td>\n<td>SU14813 maleate<\/td>\n<td>849643-15-8<\/td>\n<td>98.00%<\/td>\n<td>VEGFR\/PDGFR\/Kit\/FLT-3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3847<\/td>\n<td>SU5416<\/td>\n<td>204005-46-9<\/td>\n<td>99.06%<\/td>\n<td>VEGF receptor inhibitor and AHR agonist<\/td>\n<\/tr>\n<tr>\n<td>A3848<\/td>\n<td>Tacalcitol<\/td>\n<td>57333-96-7<\/td>\n<td>98.00%<\/td>\n<td>Promotes normal bone development by regulating calcium<\/td>\n<\/tr>\n<tr>\n<td>A3850<\/td>\n<td>TAK-242<\/td>\n<td>243984-11-4<\/td>\n<td>99.53%<\/td>\n<td>TLR 4 signaling inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3853<\/td>\n<td>Talarozole<\/td>\n<td>201410-53-9<\/td>\n<td>98.00%<\/td>\n<td>Cytochrome P450 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3854<\/td>\n<td>Talnetant<\/td>\n<td>174636-32-9<\/td>\n<td>98.00%<\/td>\n<td>NK3 receptor antagonist,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3856<\/td>\n<td>Tamibarotene<\/td>\n<td>94497-51-5<\/td>\n<td>98.41%<\/td>\n<td>RAR\u03b1 agonist<\/td>\n<\/tr>\n<tr>\n<td>A3857<\/td>\n<td>Tanaproget<\/td>\n<td>304853-42-7<\/td>\n<td>98.00%<\/td>\n<td>Progesterone receptor agonist<\/td>\n<\/tr>\n<tr>\n<td>A3858<\/td>\n<td>Taranabant<\/td>\n<td>701977-09-5<\/td>\n<td>98.00%<\/td>\n<td>Cannabinoid receptor type 1 inverse agonist<\/td>\n<\/tr>\n<tr>\n<td>A3859<\/td>\n<td>Tariquidar methanesulfonate, hydrate<\/td>\n<td>625375-83-9<\/td>\n<td>99.49%<\/td>\n<td>P-glycoprotein inhibitor, potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3860<\/td>\n<td>Tasquinimod<\/td>\n<td>254964-60-8<\/td>\n<td>99.47%<\/td>\n<td>Antiangiogenic and antineoplastic agent<\/td>\n<\/tr>\n<tr>\n<td>A3861<\/td>\n<td>TBB<\/td>\n<td>17374-26-4<\/td>\n<td>99.23%<\/td>\n<td>Casein kinase-2 (CK2) inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3862<\/td>\n<td>TC-DAPK 6<\/td>\n<td>315694-89-4<\/td>\n<td>98.00%<\/td>\n<td>DAPK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3863<\/td>\n<td>Tedizolid<\/td>\n<td>856866-72-3<\/td>\n<td>99.63%<\/td>\n<td>Oxazolidinone for gram-positive infections<\/td>\n<\/tr>\n<tr>\n<td>A3864<\/td>\n<td>Tegobuvir<\/td>\n<td>1000787-75-6<\/td>\n<td>98.97%<\/td>\n<td>HCV RNA replication inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3865<\/td>\n<td>Teneligliptin hydrobromide<\/td>\n<td>906093-29-6<\/td>\n<td>99.90%<\/td>\n<td>Dipeptidyl peptidase-4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3870<\/td>\n<td>TG 100801<\/td>\n<td>867331-82-6<\/td>\n<td>98.00%<\/td>\n<td>Multi-kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3872<\/td>\n<td>TH-302<\/td>\n<td>918633-87-1<\/td>\n<td>98.40%<\/td>\n<td>Hypoxia-activated prodrug,inhibits H460\/HT29 cell growth<\/td>\n<\/tr>\n<tr>\n<td>A3873<\/td>\n<td>Tianeptine<\/td>\n<td>66981-73-5; 72797-41-2<\/td>\n<td>99.46%<\/td>\n<td>5-HT facilitator<\/td>\n<\/tr>\n<tr>\n<td>A3874<\/td>\n<td>Tiotropium Bromide<\/td>\n<td>136310-93-5<\/td>\n<td>99.39%<\/td>\n<td>MAChR M antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3875<\/td>\n<td>Tipiracil hydrochloride<\/td>\n<td>183204-72-0<\/td>\n<td>99.74%<\/td>\n<td>Thymidine phosphorylase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3876<\/td>\n<td>Tipranavir<\/td>\n<td>174484-41-4<\/td>\n<td>98.00%<\/td>\n<td>HIV protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3877<\/td>\n<td>Tirofiban hydrochloride monohydrate<\/td>\n<td>150915-40-5<\/td>\n<td>99.46%<\/td>\n<td>Glycoprotein IIb\/IIIa inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3878<\/td>\n<td>TMC353121<\/td>\n<td>857066-90-1<\/td>\n<td>98.00%<\/td>\n<td>Potent RSV fusion inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3879<\/td>\n<td>Toceranib<\/td>\n<td>356068-94-5<\/td>\n<td>98.00%<\/td>\n<td>c-Kit\/VEGFR\/PDGFR inhibtor<\/td>\n<\/tr>\n<tr>\n<td>A3881<\/td>\n<td>Toll-like receptor modulator<\/td>\n<td>926927-42-6<\/td>\n<td>98.00%<\/td>\n<td>TLR antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3883<\/td>\n<td>Tonabersat<\/td>\n<td>175013-84-0<\/td>\n<td>98.00%<\/td>\n<td>Gap junction modulator,novel benzopyran compound for Migraine and epilepsy treatment<\/td>\n<\/tr>\n<tr>\n<td>A3884<\/td>\n<td>Toremifene<\/td>\n<td>89778-26-7<\/td>\n<td>98.00%<\/td>\n<td>Estrogen-receptor modulator<\/td>\n<\/tr>\n<tr>\n<td>A3885<\/td>\n<td>Tozadenant<\/td>\n<td>870070-55-6<\/td>\n<td>99.46%<\/td>\n<td>Adenosine 2a receptor antagonist,novel and selective<\/td>\n<\/tr>\n<tr>\n<td>A3886<\/td>\n<td>Trabectedin<\/td>\n<td>114899-77-3<\/td>\n<td>98.00%<\/td>\n<td>Antitumour agent<\/td>\n<\/tr>\n<tr>\n<td>A3887<\/td>\n<td>Trametinib DMSO solvate<\/td>\n<td>1187431-43-1<\/td>\n<td>98.64%<\/td>\n<td>Allosteric MEK1\/MEK2 kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3888<\/td>\n<td>Trelagliptin<\/td>\n<td>865759-25-7<\/td>\n<td>99.66%<\/td>\n<td>DPP-4 inhibitor,long-acting and selective<\/td>\n<\/tr>\n<tr>\n<td>A3889<\/td>\n<td>Trelagliptin succinate<\/td>\n<td>1029877-94-8<\/td>\n<td>98.00%<\/td>\n<td>DPP-4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3891<\/td>\n<td>Triptolide<\/td>\n<td>38748-32-2<\/td>\n<td>99.16%<\/td>\n<td>IL-2\/MMP-3\/MMP7\/MMP19 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3892<\/td>\n<td>Triptonide<\/td>\n<td>38647-11-9<\/td>\n<td>99.15%<\/td>\n<td>dCTP Pyrophosphatase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3893<\/td>\n<td>Troglitazone<\/td>\n<td>97322-87-7<\/td>\n<td>98.99%<\/td>\n<td>Selective PPAR\u03b3 agonist<\/td>\n<\/tr>\n<tr>\n<td>A3894<\/td>\n<td>TTP 22<\/td>\n<td>329907-28-0<\/td>\n<td>98.33%<\/td>\n<td>CK2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3895<\/td>\n<td>TUG-770<\/td>\n<td>1402601-82-4<\/td>\n<td>99.46%<\/td>\n<td>FFA1\/GPR40 agonist<\/td>\n<\/tr>\n<tr>\n<td>A3896<\/td>\n<td>Tulathromycin A<\/td>\n<td>217500-96-4<\/td>\n<td>98.00%<\/td>\n<td>Triamilide antimicrobial<\/td>\n<\/tr>\n<tr>\n<td>A3899<\/td>\n<td>UK-5099<\/td>\n<td>56396-35-1<\/td>\n<td>99.41%<\/td>\n<td>MCTs and MPC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3900<\/td>\n<td>Umeclidinium bromide<\/td>\n<td>869113-09-7<\/td>\n<td>98.74%<\/td>\n<td>MAChR antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3901<\/td>\n<td>UNC1215<\/td>\n<td>1415800-43-9<\/td>\n<td>98.55%<\/td>\n<td>Chemical probe for the methyllysine (Kme)<\/td>\n<\/tr>\n<tr>\n<td>A3902<\/td>\n<td>VAL-083<\/td>\n<td>23261-20-3<\/td>\n<td>98.00%<\/td>\n<td>Bi-functional alkylating agent<\/td>\n<\/tr>\n<tr>\n<td>A3903<\/td>\n<td>Valaciclovir<\/td>\n<td>124832-26-4<\/td>\n<td>98.00%<\/td>\n<td>Prodrug of aciclovir for herpes virus treatment<\/td>\n<\/tr>\n<tr>\n<td>A3905<\/td>\n<td>Valspodar<\/td>\n<td>121584-18-7<\/td>\n<td>96.32%<\/td>\n<td>P-glycoprotein inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3906<\/td>\n<td>Vandetanib hydrochloride<\/td>\n<td>524722-52-9<\/td>\n<td>99.92%<\/td>\n<td>VEGFR\/EGFR inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3909<\/td>\n<td>VCH-916<\/td>\n<td>1200133-34-1<\/td>\n<td>98.00%<\/td>\n<td>HCV NS5B polymerase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3915<\/td>\n<td>Vernakalant Hydrochloride<\/td>\n<td>748810-28-8<\/td>\n<td>98.00%<\/td>\n<td>Ion channel blocker,investigational antiarrhythmic<\/td>\n<\/tr>\n<tr>\n<td>A3918<\/td>\n<td>Vilazodone<\/td>\n<td>163521-12-8<\/td>\n<td>99.06%<\/td>\n<td>Combined SSRI and 5-HT1A receptor partial agonist<\/td>\n<\/tr>\n<tr>\n<td>A3919<\/td>\n<td>Vilazodone Hydrochloride<\/td>\n<td>163521-08-2<\/td>\n<td>98.38%<\/td>\n<td>Combined SSRI and 5-HT1A receptor partial agonist<\/td>\n<\/tr>\n<tr>\n<td>A3920<\/td>\n<td>Vinblastine sulfate<\/td>\n<td>143-67-9<\/td>\n<td>99.06%<\/td>\n<td>Anti-mitotic agent<\/td>\n<\/tr>\n<tr>\n<td>A3921<\/td>\n<td>Vinorelbine ditartrate<\/td>\n<td>125317-39-7<\/td>\n<td>99.06%<\/td>\n<td>Anti-mitotic chemotherapy drug<\/td>\n<\/tr>\n<tr>\n<td>A3923<\/td>\n<td>VO-Ohpic trihydrate<\/td>\n<td>476310-60-8<\/td>\n<td>98.00%<\/td>\n<td>PTEN inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3924<\/td>\n<td>Voreloxin<\/td>\n<td>175414-77-4<\/td>\n<td>98.00%<\/td>\n<td>Topo II inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3925<\/td>\n<td>Voreloxin Hydrochloride<\/td>\n<td>175519-16-1<\/td>\n<td>98.00%<\/td>\n<td>Antineoplastic naphthyridine analogue<\/td>\n<\/tr>\n<tr>\n<td>A3926<\/td>\n<td>Vortioxetine<\/td>\n<td>508233-74-7<\/td>\n<td>99.27%<\/td>\n<td>5-HT receptors antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3927<\/td>\n<td>VS-5584 (SB2343)<\/td>\n<td>1246560-33-7<\/td>\n<td>99.94%<\/td>\n<td>MTOR\/P13K inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3931<\/td>\n<td>VX-11e<\/td>\n<td>896720-20-0<\/td>\n<td>98.99%<\/td>\n<td>ERK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3932<\/td>\n<td>WAY 316606<\/td>\n<td>915759-45-4<\/td>\n<td>99.64%<\/td>\n<td>sFRP-1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3933<\/td>\n<td>WAY-100635<\/td>\n<td>162760-96-5<\/td>\n<td>99.64%<\/td>\n<td>5-HT1A receptor antagonist,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3935<\/td>\n<td>WEHI-539<\/td>\n<td>1431866-33-9<\/td>\n<td>99.23%<\/td>\n<td>Bcl-xL inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3936<\/td>\n<td>WHI-P97<\/td>\n<td>211555-05-4<\/td>\n<td>98.00%<\/td>\n<td>Janus kinase (JAK)-3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3937<\/td>\n<td>XL019<\/td>\n<td>945755-56-6<\/td>\n<td>97.66%<\/td>\n<td>JAK2 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3939<\/td>\n<td>XL228<\/td>\n<td>898280-07-4<\/td>\n<td>99.32%<\/td>\n<td>IGF1R\/AURORA \/FGFR1-3\/ABL\/SRC family kinases inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3940<\/td>\n<td>XL388<\/td>\n<td>1251156-08-7<\/td>\n<td>98.00%<\/td>\n<td>MTOR inhibitor,highly potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3942<\/td>\n<td>XMD17-109<\/td>\n<td>1435488-37-1<\/td>\n<td>99.71%<\/td>\n<td>ERK-5 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3943<\/td>\n<td>XMD8-92<\/td>\n<td>1234480-50-2<\/td>\n<td>98.18%<\/td>\n<td>BMK1\/ERK5 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3944<\/td>\n<td>X-NeuNAc<\/td>\n<td>160369-85-7<\/td>\n<td>99.58%<\/td>\n<td>Subtrate for chromogeneic assay of neuraminidase activity<\/td>\n<\/tr>\n<tr>\n<td>A3946<\/td>\n<td>YK-4-279<\/td>\n<td>1037184-44-3<\/td>\n<td>99.72%<\/td>\n<td>RNA Helicase A (RHA) inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3947<\/td>\n<td>YM-155 hydrochloride<\/td>\n<td>355406-09-6<\/td>\n<td>98.00%<\/td>\n<td>Potent survivin inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3950<\/td>\n<td>Zardaverine<\/td>\n<td>101975-10-4<\/td>\n<td>98.00%<\/td>\n<td>PDE III and IV inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3952<\/td>\n<td>Ziprasidone<\/td>\n<td>146939-27-7<\/td>\n<td>97.77%<\/td>\n<td>5-HT (serotonin)\/dopamine receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3953<\/td>\n<td>Ziprasidone hydrochloride monohydrate<\/td>\n<td>138982-67-9<\/td>\n<td>98.30%<\/td>\n<td>5-HT (serotonin)\/dopamine receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A3954<\/td>\n<td>ZM323881<\/td>\n<td>193001-14-8<\/td>\n<td>98.00%<\/td>\n<td>VEGFR-2\/KDR inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3956<\/td>\n<td>Zosuquidar<\/td>\n<td>167354-41-8<\/td>\n<td>98.49%<\/td>\n<td>MDR modulator<\/td>\n<\/tr>\n<tr>\n<td>A3958<\/td>\n<td>Veliparib dihydrochloride<\/td>\n<td>912445-05-7<\/td>\n<td>98.56%<\/td>\n<td>PARP-1\/PARP-2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3962<\/td>\n<td>AZD1208<\/td>\n<td>1204144-28-4<\/td>\n<td>99.82%<\/td>\n<td>PIM kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A3963<\/td>\n<td>A-769662<\/td>\n<td>844499-71-4<\/td>\n<td>97.68%<\/td>\n<td>AMPK activator,potent and reversible<\/td>\n<\/tr>\n<tr>\n<td>A3965<\/td>\n<td>BI 2536<\/td>\n<td>755038-02-9<\/td>\n<td>98.78%<\/td>\n<td>Plk1 inhibitor,potent and ATP-competitive<\/td>\n<\/tr>\n<tr>\n<td>A3966<\/td>\n<td>Doxorubicin<\/td>\n<td>23214-92-8<\/td>\n<td>99.31%<\/td>\n<td>Topo II inhibitor,immunosuppresive antineoplastic antibiotic<\/td>\n<\/tr>\n<tr>\n<td>A3967<\/td>\n<td>Lapatinib Ditosylate<\/td>\n<td>388082-77-7<\/td>\n<td>99.94%<\/td>\n<td>EGFR\/HER2 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3968<\/td>\n<td>PF-03716556<\/td>\n<td>928774-43-0<\/td>\n<td>98.00%<\/td>\n<td>Acid pump antagonist,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A3969<\/td>\n<td>Vatalanib<\/td>\n<td>212141-54-3<\/td>\n<td>99.57%<\/td>\n<td>VEGFR-1\/-2 inhibitor,cell-permeable<\/td>\n<\/tr>\n<tr>\n<td>A4002<\/td>\n<td>IU1<\/td>\n<td>314245-33-5<\/td>\n<td>99.00%<\/td>\n<td>Usp14 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4003<\/td>\n<td>LDN 57444<\/td>\n<td>668467-91-2<\/td>\n<td>99.79%<\/td>\n<td>UCH-L1 inhibitor,reversible competitve<\/td>\n<\/tr>\n<tr>\n<td>A4004<\/td>\n<td>NSC 632839 hydrochloride<\/td>\n<td>157654-67-6<\/td>\n<td>98.68%<\/td>\n<td>Isopeptidases inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4005<\/td>\n<td>RO4929097<\/td>\n<td>847925-91-1<\/td>\n<td>99.40%<\/td>\n<td>\u03b3 secretase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4006<\/td>\n<td>MK-0752<\/td>\n<td>471905-41-6<\/td>\n<td>99.45%<\/td>\n<td>\u03b3-secretase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4007<\/td>\n<td>MLN9708<\/td>\n<td>1201902-80-8<\/td>\n<td>99.16%<\/td>\n<td>Proteasome inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4008<\/td>\n<td>MLN2238<\/td>\n<td>1072833-77-2<\/td>\n<td>98.00%<\/td>\n<td>\u03b25 site of the 20S proteasome inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4009<\/td>\n<td>CEP-18770<\/td>\n<td>847499-27-8<\/td>\n<td>98.00%<\/td>\n<td>Proteasome inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4010<\/td>\n<td>Salinosporamide A (NPI-0052, Marizomib)<\/td>\n<td>437742-34-2<\/td>\n<td>\u226595.00%<\/td>\n<td>20S proteasome inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4011<\/td>\n<td>ONX-0914 (PR-957)<\/td>\n<td>960374-59-8<\/td>\n<td>95.30%<\/td>\n<td>Immunoproteasome inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4012<\/td>\n<td>Gabexate mesylate<\/td>\n<td>56974-61-9<\/td>\n<td>99.41%<\/td>\n<td>Trypsin-like serine proteinases inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4013<\/td>\n<td>Aspirin (Acetylsalicylic acid)<\/td>\n<td>50-78-2<\/td>\n<td>98.92%<\/td>\n<td>Cyclooxygenase (COX) inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4014<\/td>\n<td>Artemether (SM-224)<\/td>\n<td>71963-77-4<\/td>\n<td>98.00%<\/td>\n<td>Semi-synthetic derivative of artemisinin<\/td>\n<\/tr>\n<tr>\n<td>A4015<\/td>\n<td>Disulfiram<\/td>\n<td>97-77-8<\/td>\n<td>98.00%<\/td>\n<td>Dopamine \u03b2-hydroxylase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4016<\/td>\n<td>Apoptosis Activator 2<\/td>\n<td>79183-19-0<\/td>\n<td>98.00%<\/td>\n<td>Indoledione caspase activator, cell-permeable<\/td>\n<\/tr>\n<tr>\n<td>A4018<\/td>\n<td>YO-01027 (Dibenzazepine, DBZ)<\/td>\n<td>209984-56-5<\/td>\n<td>98.30%<\/td>\n<td>\u03b3-secretase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4019<\/td>\n<td>LY-411575<\/td>\n<td>209984-57-6<\/td>\n<td>98.21%<\/td>\n<td>Gamma secretase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4020<\/td>\n<td>LY2811376<\/td>\n<td>1194044-20-6<\/td>\n<td>98.00%<\/td>\n<td>Non-peptidic BACE1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4022<\/td>\n<td>BMS-708163 (Avagacestat)<\/td>\n<td>1146699-66-2<\/td>\n<td>98.73%<\/td>\n<td>\u03b3-secretase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4023<\/td>\n<td>LY3039478<\/td>\n<td>1421438-81-4<\/td>\n<td>97.16%<\/td>\n<td>Notch inhibitor, novel and potent<\/td>\n<\/tr>\n<tr>\n<td>A4024<\/td>\n<td>Danoprevir (RG7227)<\/td>\n<td>850876-88-9<\/td>\n<td>98.47%<\/td>\n<td>HCV NS3\/4A protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4031<\/td>\n<td>Telaprevir (VX-950)<\/td>\n<td>402957-28-2<\/td>\n<td>98.00%<\/td>\n<td>HCV NS3-4A protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4032<\/td>\n<td>VX-222 (VCH-222, Lomibuvir)<\/td>\n<td>1026785-59-0<\/td>\n<td>99.91%<\/td>\n<td>NNI of HCV RNA polymerase<\/td>\n<\/tr>\n<tr>\n<td>A4033<\/td>\n<td>Glimepiride<\/td>\n<td>93479-97-1<\/td>\n<td>98.14%<\/td>\n<td>Sulfonylurea compound<\/td>\n<\/tr>\n<tr>\n<td>A4034<\/td>\n<td>Linagliptin (BI-1356)<\/td>\n<td>668270-12-0<\/td>\n<td>99.69%<\/td>\n<td>DDP-4 inhibitor,highly potent and competitive<\/td>\n<\/tr>\n<tr>\n<td>A4036<\/td>\n<td>Sitagliptin phosphate monohydrate<\/td>\n<td>654671-77-9<\/td>\n<td>98.19%<\/td>\n<td>Potent DPP-4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4037<\/td>\n<td>Vildagliptin (LAF-237)<\/td>\n<td>274901-16-5<\/td>\n<td>98.05%<\/td>\n<td>DPP-4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4038<\/td>\n<td>Alogliptin (SYR-322)<\/td>\n<td>850649-61-5<\/td>\n<td>97.66%<\/td>\n<td>DPP-4 inhibitor,potent and highly selective<\/td>\n<\/tr>\n<tr>\n<td>A4040<\/td>\n<td>Atazanavir sulfate (BMS-232632-05)<\/td>\n<td>229975-97-7<\/td>\n<td>99.68%<\/td>\n<td>Protease inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4049<\/td>\n<td>Marimastat<\/td>\n<td>154039-60-8<\/td>\n<td>98.00%<\/td>\n<td>MMPs inhibitor,board spectrum<\/td>\n<\/tr>\n<tr>\n<td>A4050<\/td>\n<td>GM 6001<\/td>\n<td>142880-36-2<\/td>\n<td>98.68%<\/td>\n<td>Broad spectrum MMP inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4051<\/td>\n<td>NSC 405020<\/td>\n<td>7497-07-6<\/td>\n<td>99.13%<\/td>\n<td>MT1-MMP inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4052<\/td>\n<td>Doxycycline hyclate<\/td>\n<td>24390-14-5<\/td>\n<td>98.00%<\/td>\n<td>MMP inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4054<\/td>\n<td>17-AAG (KOS953)<\/td>\n<td>75747-14-7<\/td>\n<td>98.53%<\/td>\n<td>Hsp90 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4056<\/td>\n<td>AT13387<\/td>\n<td>912999-49-6<\/td>\n<td>99.12%<\/td>\n<td>Hsp90 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4057<\/td>\n<td>AUY922 (NVP-AUY922)<\/td>\n<td>747412-49-3<\/td>\n<td>98.26%<\/td>\n<td>Potent Hsp90 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4058<\/td>\n<td>BIIB021<\/td>\n<td>848695-25-0<\/td>\n<td>99.51%<\/td>\n<td>Hsp90 inhibitor,selective and competitive<\/td>\n<\/tr>\n<tr>\n<td>A4060<\/td>\n<td>Geldanamycin<\/td>\n<td>30562-34-6<\/td>\n<td>97.01%<\/td>\n<td>Hsp90 inhibitor,potent and specific<\/td>\n<\/tr>\n<tr>\n<td>A4061<\/td>\n<td>IPI-504 (Retaspimycin hydrochloride)<\/td>\n<td>857402-63-2<\/td>\n<td>98.20%<\/td>\n<td>Hsp90 inhibitor,novel, potent,selective<\/td>\n<\/tr>\n<tr>\n<td>A4062<\/td>\n<td>KW-2478<\/td>\n<td>819812-04-9<\/td>\n<td>98.00%<\/td>\n<td>Potent Hsp90 inhibitor, novel, non-ansamycin,<\/td>\n<\/tr>\n<tr>\n<td>A4063<\/td>\n<td>MPC-3100<\/td>\n<td>958025-66-6<\/td>\n<td>98.00%<\/td>\n<td>Hsp90 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4064<\/td>\n<td>NVP-BEP800<\/td>\n<td>847559-80-2<\/td>\n<td>99.22%<\/td>\n<td>Oral Hsp90\u03b2 inhibitor, novel, fully synthetic<\/td>\n<\/tr>\n<tr>\n<td>A4065<\/td>\n<td>PF-04929113 (SNX-5422)<\/td>\n<td>908115-27-5<\/td>\n<td>99.61%<\/td>\n<td>Hsp90 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4067<\/td>\n<td>Radicicol<\/td>\n<td>12772-57-5<\/td>\n<td>98.00%<\/td>\n<td>ATPase\/kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4068<\/td>\n<td>SNX-2112<\/td>\n<td>908112-43-6<\/td>\n<td>98.00%<\/td>\n<td>Hsp90 inhibitor,ATP-competitve,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4069<\/td>\n<td>BMS-707035<\/td>\n<td>729607-74-3<\/td>\n<td>99.68%<\/td>\n<td>HIV-I integrase inhibitor,potent and specific<\/td>\n<\/tr>\n<tr>\n<td>A4070<\/td>\n<td>Elvitegravir (GS-9137)<\/td>\n<td>697761-98-1<\/td>\n<td>99.07%<\/td>\n<td>HIV-1 integrase inhibitor,potent<\/td>\n<\/tr>\n<tr>\n<td>A4071<\/td>\n<td>Fluorouracil (Adrucil)<\/td>\n<td>51-21-8<\/td>\n<td>99.94%<\/td>\n<td>Antitumor agent;inhibitor of thymidylate synthase<\/td>\n<\/tr>\n<tr>\n<td>A4073<\/td>\n<td>Raltegravir (MK-0518)<\/td>\n<td>518048-05-0<\/td>\n<td>99.73%<\/td>\n<td>HIV-1 integrase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4074<\/td>\n<td>S\/GSK1349572<\/td>\n<td>1051375-16-6<\/td>\n<td>99.89%<\/td>\n<td>HIV integrase inhibitor, novel and potent<\/td>\n<\/tr>\n<tr>\n<td>A4077<\/td>\n<td>BIBR 953 (Dabigatran, Pradaxa)<\/td>\n<td>211914-51-1<\/td>\n<td>99.44%<\/td>\n<td>Thrombin inhibitor,potent,reversible and direct<\/td>\n<\/tr>\n<tr>\n<td>A4078<\/td>\n<td>Captopril<\/td>\n<td>62571-86-2<\/td>\n<td>98.91%<\/td>\n<td>ACE inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4079<\/td>\n<td>Fosinopril sodium<\/td>\n<td>88889-14-9<\/td>\n<td>98.00%<\/td>\n<td>ACE inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4080<\/td>\n<td>Moxonidine<\/td>\n<td>75438-57-2<\/td>\n<td>99.53%<\/td>\n<td>I1R\/\u03b12AR agonist<\/td>\n<\/tr>\n<tr>\n<td>A4082<\/td>\n<td>Olmesartan medoxomil<\/td>\n<td>144689-63-4<\/td>\n<td>99.38%<\/td>\n<td>AT1 receptor antagonist<\/td>\n<\/tr>\n<tr>\n<td>A4083<\/td>\n<td>Rocilinostat (ACY-1215)<\/td>\n<td>1316214-52-4<\/td>\n<td>99.40%<\/td>\n<td>Selective HDAC6 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4084<\/td>\n<td>Vorinostat (SAHA, MK0683)<\/td>\n<td>149647-78-9<\/td>\n<td>99.89%<\/td>\n<td>HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4089<\/td>\n<td>Mocetinostat (MGCD0103, MG0103)<\/td>\n<td>726169-73-9<\/td>\n<td>98.49%<\/td>\n<td>HDAC inhibitor,isotype-selective and potent<\/td>\n<\/tr>\n<tr>\n<td>A4090<\/td>\n<td>JNJ-26481585<\/td>\n<td>875320-29-9<\/td>\n<td>99.01%<\/td>\n<td>Potent HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4091<\/td>\n<td>PCI-34051<\/td>\n<td>950762-95-5<\/td>\n<td>98.67%<\/td>\n<td>HDAC8 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4092<\/td>\n<td>CUDC-101<\/td>\n<td>1012054-59-9<\/td>\n<td>99.56%<\/td>\n<td>Multitargeted HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4093<\/td>\n<td>ITF2357 (Givinostat)<\/td>\n<td>732302-99-7<\/td>\n<td>98.28%<\/td>\n<td>HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4094<\/td>\n<td>MC1568<\/td>\n<td>852475-26-4<\/td>\n<td>98.44%<\/td>\n<td>Class II HDAC inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4095<\/td>\n<td>Pracinostat (SB939)<\/td>\n<td>929016-96-6<\/td>\n<td>98.89%<\/td>\n<td>Pan-HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4096<\/td>\n<td>Belinostat (PXD101)<\/td>\n<td>414864-00-9<\/td>\n<td>98.04%<\/td>\n<td>Hydroxamate-type HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4097<\/td>\n<td>CUDC-907<\/td>\n<td>1339928-25-4<\/td>\n<td>98.06%<\/td>\n<td>Potent PI3K\/HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4098<\/td>\n<td>PCI-24781 (CRA-024781)<\/td>\n<td>783355-60-2<\/td>\n<td>98.01%<\/td>\n<td>Pan-HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4099<\/td>\n<td>Valproic acid sodium salt (Sodium valproate)<\/td>\n<td>1069-66-5<\/td>\n<td>98.07%<\/td>\n<td>HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4100<\/td>\n<td>Droxinostat<\/td>\n<td>99873-43-5<\/td>\n<td>98.00%<\/td>\n<td>Selective HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4101<\/td>\n<td>Tubastatin A<\/td>\n<td>1252003-15-8<\/td>\n<td>98.00%<\/td>\n<td>HDAC6 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4102<\/td>\n<td>CI994 (Tacedinaline)<\/td>\n<td>112522-64-2<\/td>\n<td>98.17%<\/td>\n<td>HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4103<\/td>\n<td>LAQ824 (NVP-LAQ824,Dacinostat)<\/td>\n<td>404951-53-7<\/td>\n<td>98.12%<\/td>\n<td>HDAC inhibitor,potent and novel<\/td>\n<\/tr>\n<tr>\n<td>A4104<\/td>\n<td>AR-42 (OSU-HDAC42)<\/td>\n<td>935881-37-1<\/td>\n<td>99.03%<\/td>\n<td>HDAC inhibitor,novel and potent<\/td>\n<\/tr>\n<tr>\n<td>A4105<\/td>\n<td>M344<\/td>\n<td>251456-60-7<\/td>\n<td>98.73%<\/td>\n<td>HDAC inhibitor,potent and cell-permeable<\/td>\n<\/tr>\n<tr>\n<td>A4106<\/td>\n<td>Scriptaid<\/td>\n<td>287383-59-9<\/td>\n<td>98.70%<\/td>\n<td>HDAC inhibitor,novel and cell-permeable<\/td>\n<\/tr>\n<tr>\n<td>A4107<\/td>\n<td>Sodium Phenylbutyrate<\/td>\n<td>1716-12-7<\/td>\n<td>99.78%<\/td>\n<td>Histone deacetylase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4108<\/td>\n<td>Resminostat (RAS2410)<\/td>\n<td>864814-88-0<\/td>\n<td>98.00%<\/td>\n<td>Potent HDAC inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4110<\/td>\n<td>MLN8237 (Alisertib)<\/td>\n<td>1028486-01-2<\/td>\n<td>98.77%<\/td>\n<td>Aurora A Kinase inhibitor, Potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4111<\/td>\n<td>VX-680 (MK-0457,Tozasertib)<\/td>\n<td>639089-54-6<\/td>\n<td>99.93%<\/td>\n<td>Aurora kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4112<\/td>\n<td>Barasertib (AZD1152-HQPA)<\/td>\n<td>722544-51-6<\/td>\n<td>98.25%<\/td>\n<td>Aurora Kinase B inhibitor, Potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4113<\/td>\n<td>ZM 447439<\/td>\n<td>331771-20-1<\/td>\n<td>98.80%<\/td>\n<td>Aurora Kinase inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4114<\/td>\n<td>MLN8054<\/td>\n<td>869363-13-3<\/td>\n<td>97.64%<\/td>\n<td>Aurora A inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4115<\/td>\n<td>JNJ-7706621<\/td>\n<td>443797-96-4<\/td>\n<td>98.11%<\/td>\n<td>Potent CDK\/Aurora kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4116<\/td>\n<td>Danusertib (PHA-739358)<\/td>\n<td>827318-97-8<\/td>\n<td>99.39%<\/td>\n<td>Pan-aurora kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4117<\/td>\n<td>AT9283<\/td>\n<td>896466-04-9<\/td>\n<td>99.29%<\/td>\n<td>Aurora kinase\/JAK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4118<\/td>\n<td>Hesperadin<\/td>\n<td>422513-13-1<\/td>\n<td>98.29%<\/td>\n<td>Aurora B kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4119<\/td>\n<td>AMG-900<\/td>\n<td>945595-80-2<\/td>\n<td>98.99%<\/td>\n<td>Aurora kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4120<\/td>\n<td>MK-5108 (VX-689)<\/td>\n<td>1010085-13-8<\/td>\n<td>96.91%<\/td>\n<td>Aurora-A kinase inhibitor,highly selective<\/td>\n<\/tr>\n<tr>\n<td>A4121<\/td>\n<td>SNS-314 Mesylate<\/td>\n<td>1146618-41-8<\/td>\n<td>99.94%<\/td>\n<td>Aurora A\/B\/C kinases inhibitor, potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4122<\/td>\n<td>PHA-680632<\/td>\n<td>398493-79-3<\/td>\n<td>98.53%<\/td>\n<td>Aurora kinase inhibitor,novel and potent<\/td>\n<\/tr>\n<tr>\n<td>A4123<\/td>\n<td>KW 2449<\/td>\n<td>1000669-72-6<\/td>\n<td>99.94%<\/td>\n<td>Multikinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4124<\/td>\n<td>TAK-901<\/td>\n<td>934541-31-8<\/td>\n<td>98.00%<\/td>\n<td>Novel Aurora A\/B inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4125<\/td>\n<td>CYC116<\/td>\n<td>693228-63-6<\/td>\n<td>98.71%<\/td>\n<td>Potent Aurora A\/B inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4126<\/td>\n<td>Aurora A Inhibitor I<\/td>\n<td>1158838-45-9<\/td>\n<td>98.83%<\/td>\n<td>Aurora A inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4127<\/td>\n<td>GSK1070916<\/td>\n<td>942918-07-2<\/td>\n<td>98.00%<\/td>\n<td>Aurora B\/C inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4128<\/td>\n<td>PF-03814735<\/td>\n<td>942487-16-3<\/td>\n<td>98.00%<\/td>\n<td>Aurora A\/B inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4129<\/td>\n<td>ENMD-2076 L-(+)-Tartaric acid<\/td>\n<td>1291074-87-7<\/td>\n<td>99.36%<\/td>\n<td>Aurora kinases inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4130<\/td>\n<td>ENMD-2076<\/td>\n<td>934353-76-1<\/td>\n<td>98.78%<\/td>\n<td>Selective Aurora A\/Flt3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4132<\/td>\n<td>CCT137690<\/td>\n<td>1095382-05-0<\/td>\n<td>98.00%<\/td>\n<td>Aurora A\/B\/C inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4135<\/td>\n<td>Tofacitinib (CP-690550) Citrate<\/td>\n<td>540737-29-9<\/td>\n<td>99.64%<\/td>\n<td>Potent JAK inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4136<\/td>\n<td>TG101348 (SAR302503)<\/td>\n<td>936091-26-8<\/td>\n<td>99.39%<\/td>\n<td>JAK-2 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4137<\/td>\n<td>AZD1480<\/td>\n<td>935666-88-9<\/td>\n<td>99.31%<\/td>\n<td>JAK2 inhibitor,ATP-competitive and novel<\/td>\n<\/tr>\n<tr>\n<td>A4138<\/td>\n<td>Tofacitinib (CP-690550,Tasocitinib)<\/td>\n<td>477600-75-2<\/td>\n<td>99.94%<\/td>\n<td>Janus kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4139<\/td>\n<td>AG-490<\/td>\n<td>133550-30-8<\/td>\n<td>99.76%<\/td>\n<td>JAK2\/EGFR inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4140<\/td>\n<td>WP1066<\/td>\n<td>857064-38-1<\/td>\n<td>99.84%<\/td>\n<td>JAK2\/STAT3 inhibitor,cell-permeable<\/td>\n<\/tr>\n<tr>\n<td>A4141<\/td>\n<td>Baricitinib (LY3009104, INCB028050)<\/td>\n<td>1187594-09-7<\/td>\n<td>98.06%<\/td>\n<td>JAK1\/JAK2 inhibitor,selective orally bioavailable<\/td>\n<\/tr>\n<tr>\n<td>A4143<\/td>\n<td>CYT387<\/td>\n<td>1056634-68-4<\/td>\n<td>98.70%<\/td>\n<td>JAK-1\/-2 inhibitor,ATP competitive<\/td>\n<\/tr>\n<tr>\n<td>A4144<\/td>\n<td>AZ 960<\/td>\n<td>905586-69-8<\/td>\n<td>98.00%<\/td>\n<td>JAKs inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4145<\/td>\n<td>TG101209<\/td>\n<td>936091-14-4<\/td>\n<td>99.46%<\/td>\n<td>JAK2\/3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4146<\/td>\n<td>CEP-33779<\/td>\n<td>1257704-57-6<\/td>\n<td>98.00%<\/td>\n<td>JAK2 inhibitor,highly selective<\/td>\n<\/tr>\n<tr>\n<td>A4147<\/td>\n<td>LY2784544<\/td>\n<td>1229236-86-5<\/td>\n<td>98.00%<\/td>\n<td>JAK2 inhibitor,highly potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4148<\/td>\n<td>NVP-BSK805 2HCl<\/td>\n<td>1092499-93-8 (free base)<\/td>\n<td>99.23%<\/td>\n<td>JAK2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4149<\/td>\n<td>S-Ruxolitinib (INCB018424)<\/td>\n<td>941685-37-6<\/td>\n<td>99.34%<\/td>\n<td>JAK1\/2 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4150<\/td>\n<td>WHI-P154<\/td>\n<td>211555-04-3<\/td>\n<td>99.19%<\/td>\n<td>JAK3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4151<\/td>\n<td>ZM 39923 HCl<\/td>\n<td>1021868-92-7<\/td>\n<td>99.91%<\/td>\n<td>JAK3 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4152<\/td>\n<td>BMS-911543<\/td>\n<td>1271022-90-2<\/td>\n<td>98.41%<\/td>\n<td>JAK2 inhibitor,selective small molecule<\/td>\n<\/tr>\n<tr>\n<td>A4153<\/td>\n<td>BMN 673<\/td>\n<td>1207456-01-6<\/td>\n<td>99.26%<\/td>\n<td>Potent PARP inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4154<\/td>\n<td>Olaparib (AZD2281, Ku-0059436)<\/td>\n<td>763113-22-0<\/td>\n<td>99.80%<\/td>\n<td>Potent PARP1\/PARP2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4156<\/td>\n<td>Rucaparib (AG-014699,PF-01367338)<\/td>\n<td>459868-92-9<\/td>\n<td>98.46%<\/td>\n<td>Potent PARP inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4157<\/td>\n<td>Iniparib (BSI-201)<\/td>\n<td>160003-66-7<\/td>\n<td>99.08%<\/td>\n<td>PARP1 inhibitor,intravenously adminsitered<\/td>\n<\/tr>\n<tr>\n<td>A4158<\/td>\n<td>AG-14361<\/td>\n<td>328543-09-5<\/td>\n<td>99.17%<\/td>\n<td>Potent PARP1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4159<\/td>\n<td>PJ34 hydrochloride<\/td>\n<td>344458-15-7<\/td>\n<td>99.54%<\/td>\n<td>PARP inhibitor,potent and cell-permeable<\/td>\n<\/tr>\n<tr>\n<td>A4160<\/td>\n<td>A-966492<\/td>\n<td>934162-61-5<\/td>\n<td>99.03%<\/td>\n<td>PARP-1\/-2 inhibitor, highly potent<\/td>\n<\/tr>\n<tr>\n<td>A4161<\/td>\n<td>3-aminobenzamide<\/td>\n<td>3544-24-9<\/td>\n<td>99.66%<\/td>\n<td>Potent PARP inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4163<\/td>\n<td>UPF 1069<\/td>\n<td>1048371-03-4<\/td>\n<td>98.00%<\/td>\n<td>Selective PARP2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4164<\/td>\n<td>AZD2461<\/td>\n<td>1174043-16-3<\/td>\n<td>98.00%<\/td>\n<td>Novel PARP inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4166<\/td>\n<td>EPZ5676<\/td>\n<td>1380288-87-8<\/td>\n<td>99.28%<\/td>\n<td>DOT1L inhibitor,potent and SAM competitive<\/td>\n<\/tr>\n<tr>\n<td>A4167<\/td>\n<td>SGC 0946<\/td>\n<td>1561178-17-3<\/td>\n<td>99.65%<\/td>\n<td>DOT1L inhibitor,highly potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4168<\/td>\n<td>Entacapone<\/td>\n<td>130929-57-6<\/td>\n<td>99.28%<\/td>\n<td>COMT inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4170<\/td>\n<td>EPZ004777<\/td>\n<td>1338466-77-5<\/td>\n<td>99.43%<\/td>\n<td>DOT1L inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4171<\/td>\n<td>EPZ005687<\/td>\n<td>1396772-26-1<\/td>\n<td>98.66%<\/td>\n<td>EZH2 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4176<\/td>\n<td>Thioguanine<\/td>\n<td>154-42-7<\/td>\n<td>98.18%<\/td>\n<td>Purine antimetabolite<\/td>\n<\/tr>\n<tr>\n<td>A4180<\/td>\n<td>SRT1720 HCl<\/td>\n<td>1001645-58-4<\/td>\n<td>99.52%<\/td>\n<td>SIRT1 activator<\/td>\n<\/tr>\n<tr>\n<td>A4181<\/td>\n<td>EX 527 (SEN0014196)<\/td>\n<td>49843-98-3<\/td>\n<td>99.71%<\/td>\n<td>SIRT1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4182<\/td>\n<td>Resveratrol<\/td>\n<td>501-36-0<\/td>\n<td>99.94%<\/td>\n<td>SIRT1 activator<\/td>\n<\/tr>\n<tr>\n<td>A4183<\/td>\n<td>Sirtinol<\/td>\n<td>410536-97-9<\/td>\n<td>98.00%<\/td>\n<td>SIRT inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4184<\/td>\n<td>PFI-1 (PF-6405761)<\/td>\n<td>1403764-72-6<\/td>\n<td>97.20%<\/td>\n<td>BET inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4186<\/td>\n<td>Bromosporine<\/td>\n<td>1619994-69-2<\/td>\n<td>98.00%<\/td>\n<td>Bromodomain inhibitor,non-selective<\/td>\n<\/tr>\n<tr>\n<td>A4187<\/td>\n<td>FG-4592 (ASP1517)<\/td>\n<td>808118-40-3<\/td>\n<td>99.92%<\/td>\n<td>HIF prolyl-hydroxylase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4188<\/td>\n<td>2-Methoxyestradiol (2-MeOE2)<\/td>\n<td>362-07-2<\/td>\n<td>99.00%<\/td>\n<td>Apoptotic, antiproliferative and antiangiogenic agent<\/td>\n<\/tr>\n<tr>\n<td>A4189<\/td>\n<td>IOX2(Glycine)<\/td>\n<td>931398-72-0<\/td>\n<td>98.10%<\/td>\n<td>HIF-1\u03b1 prolyl hydroxylase-2 (PHD2) inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4190<\/td>\n<td>GSK J4 HCl<\/td>\n<td>1373423-53-0(free base)<\/td>\n<td>98.00%<\/td>\n<td>Inhibitor of H3K27 demethylase JMJD3,potent and cell-permeable<\/td>\n<\/tr>\n<tr>\n<td>A4191<\/td>\n<td>GSK J1<\/td>\n<td>1373422-53-7<\/td>\n<td>99.50%<\/td>\n<td>H3K27 demethylase JMJD3 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4192<\/td>\n<td>SGI-1776 free base<\/td>\n<td>1025065-69-3<\/td>\n<td>99.19%<\/td>\n<td>Pim kinase inhibitor,ATP-competitive<\/td>\n<\/tr>\n<tr>\n<td>A4193<\/td>\n<td>SMI-4a<\/td>\n<td>438190-29-5<\/td>\n<td>99.76%<\/td>\n<td>Potent Pim inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4194<\/td>\n<td>Obatoclax mesylate (GX15-070)<\/td>\n<td>803712-79-0<\/td>\n<td>98.49%<\/td>\n<td>Potent Bcl-2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4199<\/td>\n<td>Sabutoclax<\/td>\n<td>1228108-65-3<\/td>\n<td>98.00%<\/td>\n<td>pan-Bcl-2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4200<\/td>\n<td>Apogossypolone (ApoG2)<\/td>\n<td>886578-07-0<\/td>\n<td>98.00%<\/td>\n<td>Bcl-2 inhibitor,nonpeptidic small molecule<\/td>\n<\/tr>\n<tr>\n<td>A4202<\/td>\n<td>RITA (NSC 652287)<\/td>\n<td>213261-59-7<\/td>\n<td>99.53%<\/td>\n<td>Mdm2-p53 interaction and p53 ubiquitination blocking<\/td>\n<\/tr>\n<tr>\n<td>A4203<\/td>\n<td>Tenovin-1<\/td>\n<td>380315-80-0<\/td>\n<td>99.90%<\/td>\n<td>SIRT2 inhibitor, activates p53<\/td>\n<\/tr>\n<tr>\n<td>A4204<\/td>\n<td>JNJ-26854165 (Serdemetan)<\/td>\n<td>881202-45-5<\/td>\n<td>98.35%<\/td>\n<td>P53 activator, blocking Mdm2-p53 interaction<\/td>\n<\/tr>\n<tr>\n<td>A4206<\/td>\n<td>Pifithrin-\u03b1 (PFT\u03b1)<\/td>\n<td>63208-82-2<\/td>\n<td>98.16%<\/td>\n<td>p53 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4208<\/td>\n<td>NSC 319726<\/td>\n<td>71555-25-4<\/td>\n<td>98.00%<\/td>\n<td>Reactivator of mutant p53<\/td>\n<\/tr>\n<tr>\n<td>A4209<\/td>\n<td>NSC 207895 (XI-006)<\/td>\n<td>58131-57-0<\/td>\n<td>98.00%<\/td>\n<td>MDMX inhibitor,anti-cancer agent<\/td>\n<\/tr>\n<tr>\n<td>A4210<\/td>\n<td>Bay 11-7821 (BAY 11-7082)<\/td>\n<td>19542-67-7<\/td>\n<td>99.91%<\/td>\n<td>IKK\/NF-\u03baB\/TNF\u03b1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4211<\/td>\n<td>Lenalidomide (CC-5013)<\/td>\n<td>191732-72-6<\/td>\n<td>98.66%<\/td>\n<td>Antineoplastic agent,inhibits angiogenesis<\/td>\n<\/tr>\n<tr>\n<td>A4212<\/td>\n<td>Pomalidomide (CC-4047)<\/td>\n<td>19171-19-8<\/td>\n<td>98.46%<\/td>\n<td>Immunomodulator,antumor\/anti-angiogenic<\/td>\n<\/tr>\n<tr>\n<td>A4213<\/td>\n<td>Necrostatin-1<\/td>\n<td>4311-88-0<\/td>\n<td>99.88%<\/td>\n<td>RIP1 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4216<\/td>\n<td>Thalidomide<\/td>\n<td>50-35-1<\/td>\n<td>99.21%<\/td>\n<td>Immunomodulatory agent,sedative drug,angiogenesis inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4217<\/td>\n<td>QNZ (EVP4593)<\/td>\n<td>545380-34-5<\/td>\n<td>99.41%<\/td>\n<td>Potent NF-\u03baB inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4219<\/td>\n<td>Birinapant (TL32711)<\/td>\n<td>1260251-31-7<\/td>\n<td>98.13%<\/td>\n<td>Potent XIAP\/cIAP1 antagonist<\/td>\n<\/tr>\n<tr>\n<td>A4221<\/td>\n<td>YM155<\/td>\n<td>781661-94-7<\/td>\n<td>99.60%<\/td>\n<td>Survivin suppressant,apoptosis inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4224<\/td>\n<td>GDC-0152<\/td>\n<td>873652-48-3<\/td>\n<td>99.00%<\/td>\n<td>IAP antagonist,potent amd samll-molecule<\/td>\n<\/tr>\n<tr>\n<td>A4227<\/td>\n<td>Tipifarnib (Zarnestra)<\/td>\n<td>192185-72-1<\/td>\n<td>99.18%<\/td>\n<td>Farnesyltransferase inhibitor,potent and specific<\/td>\n<\/tr>\n<tr>\n<td>A4228<\/td>\n<td>Nutlin-3<\/td>\n<td>890090-75-2<\/td>\n<td>98.35%<\/td>\n<td>MDM2 antagonist,inhibits MDM2-p53 interaction<\/td>\n<\/tr>\n<tr>\n<td>A4230<\/td>\n<td>NSC 66811<\/td>\n<td>6964-62-1<\/td>\n<td>98.00%<\/td>\n<td>MDM2 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4232<\/td>\n<td>Cyclophosphamide monohydrate<\/td>\n<td>6055-19-2<\/td>\n<td>98.00%<\/td>\n<td>alkylating, cytotoxic agent,antitumor activity<\/td>\n<\/tr>\n<tr>\n<td>A4233<\/td>\n<td>Methylprednisolone<\/td>\n<td>83-43-2<\/td>\n<td>99.31%<\/td>\n<td>Apoptosis inducer,GR agonist<\/td>\n<\/tr>\n<tr>\n<td>A4234<\/td>\n<td>TW-37<\/td>\n<td>877877-35-5<\/td>\n<td>98.13%<\/td>\n<td>Bcl-2 inhibitor, inhibits Bcl-2,Bcl-XL and Mcl-1<\/td>\n<\/tr>\n<tr>\n<td>A4237<\/td>\n<td>Amuvatinib (MP-470, HPK 56)<\/td>\n<td>850879-09-3<\/td>\n<td>99.91%<\/td>\n<td>Tyrosine kinase inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4240<\/td>\n<td>Abiraterone<\/td>\n<td>154229-19-3<\/td>\n<td>99.30%<\/td>\n<td>Potent CYP17 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4300<\/td>\n<td>GW9662<\/td>\n<td>22978-25-2<\/td>\n<td>99.25%<\/td>\n<td>PPAR\u03b3 antagonist<\/td>\n<\/tr>\n<tr>\n<td>A4301<\/td>\n<td>T0070907<\/td>\n<td>313516-66-4<\/td>\n<td>99.88%<\/td>\n<td>Human PPAR\u03b3 antagonist,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4302<\/td>\n<td>Rosiglitazone maleate<\/td>\n<td>155141-29-0<\/td>\n<td>99.15%<\/td>\n<td>PPAR\u03b3 agonist,high-affinity and selective,potent insulin sensitizer<\/td>\n<\/tr>\n<tr>\n<td>A4303<\/td>\n<td>GSK3787<\/td>\n<td>188591-46-0<\/td>\n<td>99.73%<\/td>\n<td>PPAR\u03b2\/\u03b4 antagonist,novel and irreversible<\/td>\n<\/tr>\n<tr>\n<td>A4304<\/td>\n<td>Rosiglitazone<\/td>\n<td>122320-73-4<\/td>\n<td>99.80%<\/td>\n<td>Potent PPAR\u03b3 agonist<\/td>\n<\/tr>\n<tr>\n<td>A4305<\/td>\n<td>WY-14643 (Pirinixic Acid)<\/td>\n<td>50892-23-4<\/td>\n<td>99.87%<\/td>\n<td>PPAR\u03b1 agonist,selective and highly potent<\/td>\n<\/tr>\n<tr>\n<td>A4306<\/td>\n<td>Ciprofibrate<\/td>\n<td>52214-84-3<\/td>\n<td>98.88%<\/td>\n<td>PPAR\u03b1 agonist<\/td>\n<\/tr>\n<tr>\n<td>A4307<\/td>\n<td>GW0742<\/td>\n<td>317318-84-6<\/td>\n<td>99.64%<\/td>\n<td>PPAR\u03b4\/\u03b2 agonist,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4308<\/td>\n<td>Alizarin<\/td>\n<td>72-48-0<\/td>\n<td>98.03%<\/td>\n<td>Chelator for calcium,used to stain calcium deposites,Alizarin complexone is used for bone staining to study bone remodeling<\/td>\n<\/tr>\n<tr>\n<td>A4309<\/td>\n<td>GW501516<\/td>\n<td>317318-70-0<\/td>\n<td>98.27%<\/td>\n<td>PPAR\u03b4 agonist,selective and potent<\/td>\n<\/tr>\n<tr>\n<td>A4310<\/td>\n<td>Rosiglitazone HCl<\/td>\n<td>302543-62-0<\/td>\n<td>99.31%<\/td>\n<td>PPAR\u03b3 agonist<\/td>\n<\/tr>\n<tr>\n<td>A4311<\/td>\n<td>PF-4981517<\/td>\n<td>1390637-82-7<\/td>\n<td>98.00%<\/td>\n<td>CYP3A4 inhibitor,potent and selective<\/td>\n<\/tr>\n<tr>\n<td>A4313<\/td>\n<td>Cobicistat (GS-9350)<\/td>\n<td>1004316-88-4<\/td>\n<td>99.94%<\/td>\n<td>Selective CYP3A inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4316<\/td>\n<td>Ketoconazole<\/td>\n<td>65277-42-1<\/td>\n<td>99.48%<\/td>\n<td>Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase<\/td>\n<\/tr>\n<tr>\n<td>A4317<\/td>\n<td>Apremilast (CC-10004)<\/td>\n<td>608141-41-9<\/td>\n<td>98.98%<\/td>\n<td>PDE4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4318<\/td>\n<td>Avasimibe<\/td>\n<td>166518-60-1<\/td>\n<td>99.66%<\/td>\n<td>ACAT inhibitor,orally bioavailable<\/td>\n<\/tr>\n<tr>\n<td>A4319<\/td>\n<td>Roflumilast<\/td>\n<td>162401-32-3<\/td>\n<td>99.08%<\/td>\n<td>PDE-4 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4320<\/td>\n<td>Voriconazole<\/td>\n<td>137234-62-9<\/td>\n<td>99.96%<\/td>\n<td>CYP51 inhibitor<\/td>\n<\/tr>\n<tr>\n<td>A4321<\/td>\n<td>Sildenafil Citrate<\/td>\n<td>171599-83-0<\/td>\n<td>99.63%<\/td>\n<td>Treat erectile dysfunction and PAH<\/td>\n<\/tr>\n<tr>\n<td>A4322<\/td>\n<td>Clarithromycin<\/td>\n<td>81103-11-9<\/td>\n<td>99.39%<\/td>\n<td>CYP3A inhibitor, potent<\/td>\n<\/tr>\n<tr>\n<td>A4323<\/td>\n<td>Vardenafil HCl Trihydrate<\/td>\n<td>330808-88-3<\/td>\n<td>99.63%<\/td>\n<td>PDE5 inhibitor, potent and selective<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>\u03b2-\u5167\u91af\u80fa\u985e\u6297\u751f\u7d20\u7cfb\u5217\u5546\u54c1-&gt;&gt;\u5b89\u6bd4\u897f\u6797Ampicillin sodium APExBIO Tec [&hellip;]<\/p>\n","protected":false},"author":3,"featured_media":34209,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":[],"categories":[5368,486],"tags":[4949],"_links":{"self":[{"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/posts\/34208"}],"collection":[{"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/posts"}],"about":[{"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/types\/post"}],"author":[{"embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/users\/3"}],"replies":[{"embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=%2Fwp%2Fv2%2Fcomments&post=34208"}],"version-history":[{"count":7,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/posts\/34208\/revisions"}],"predecessor-version":[{"id":53716,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/posts\/34208\/revisions\/53716"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/media\/34209"}],"wp:attachment":[{"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=34208"}],"wp:term":[{"taxonomy":"category","embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=%2Fwp%2Fv2%2Fcategories&post=34208"},{"taxonomy":"post_tag","embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=%2Fwp%2Fv2%2Ftags&post=34208"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}