{"id":34010,"date":"2022-09-06T14:19:40","date_gmt":"2022-09-06T06:19:40","guid":{"rendered":"http:\/\/biopioneer.com.tw\/?p=34010"},"modified":"2025-06-30T18:47:47","modified_gmt":"2025-06-30T10:47:47","slug":"ms023-type-i-prmts-inhibitor%e6%8a%91%e5%88%b6%e5%8a%91-cas-1831110-54-3apexbio%e8%b2%a8%e8%99%9f-b6183","status":"publish","type":"post","link":"https:\/\/biopioneer.com.tw\/?p=34010","title":{"rendered":"MS023 (type I PRMTs inhibitor\u6291\u5236\u5291) | CAS# 1831110-54-3APExBIO\u8ca8\u865f B6183"},"content":{"rendered":"<p><strong><span style=\"font-size: 12pt; color: #ff6600;\"><span style=\"font-size: 14pt;\"><span style=\"color: #800080;\">PRMTs \u6291\u5236\u5291\u7cfb\u5217\u5546\u54c1-&gt;&gt;<span style=\"color: #ff6600;\">MS023<\/span><\/span><\/span><\/span><\/strong><\/p>\n<p>APExBIO Technology LLC \u662f\u4e00\u5bb6\u9818\u5148\u7684\u5c0f\u5206\u5b50\u6291\u5236\u5291 (Small Molecule Inhibitors)\/\u6d3b\u5316\u5291(Activators)\u3001\u5316\u5408\u7269\u5eab( Compound Libraries)\u3001\u80dc\u80bd(Peptides)\u3001\u6aa2\u6e2c\u8a66\u5291\u76d2(Assay Kits)\u3001\u87a2\u5149\u6a19\u8a18(Fluorescent Label)\u3001\u9176(Enzymes)\u3001\u4fee\u98fe\u6838\u82f7\u9178(Modified Nucleotides)\u3001mRNA \u5408\u6210\u4ee5\u53ca\u5404\u7a2e\u5206\u5b50\u751f\u7269\u5b78\u5de5\u5177\u7684\u4f9b\u61c9\u5546\u3002APExBIO\u63d0\u4f9b\u5ee3\u6cdb\u7684\u7522\u54c1\u7dda\uff0c\u6db5\u84cb 20 \u591a\u500b\u4e0d\u540c\u7684\u7814\u7a76\u9818\u57df\uff0c\u4f8b\u5982\u764c\u75c7(cancer)\u3001\u514d\u75ab\u5b78(immunology)\u3001\u795e\u7d93\u79d1\u5b78(neurosciences)\u3001\u7d30\u80de\u51cb\u4ea1(apoptosis)\u548c\u8868\u89c0\u907a\u50b3\u5b78(epigenetics)\u7b49\u3002\u516c\u53f8\u7e3d\u90e8\u4f4d\u65bc\u7f8e\u570b\u5fb7\u5dde\u4f11\u58eb\u9813USA (Houston, Texas)\uff0c\u81f4\u529b\u65bc\u670d\u52d9\u5168\u7403\u5ba2\u6236\u3002\u9ad8\u5ea6\u91cd\u8996\u7522\u54c1\u54c1\u8cea\u3002\u6240\u6709\u7522\u54c1\u5747\u9075\u5faa\u56b4\u683c\u7684\u751f\u7522\u6307\u5357\uff0c\u4e26\u9644\u6709\u5206\u6790\u8b49\u66f8\u3001HPLC\u3001\u8cea\u8b5c(Mass Spectrum)\u548cHMNR\u4ee5\u53ca\u9ad4\u5916\u9a57\u8b49(in vitro validation)\u3002 APExBIO\u7522\u54c1\u5df2\u88ab\u300aNature\u300b\u3001\u300aCell\u300b\u548c\u300aScience\u300b\u7b49\u773e\u591a\u9802\u7d1a\u540c\u884c\u8a55\u5be9\u671f\u520a\u5f15\u7528\u3002<\/p>\n<p><img decoding=\"async\" loading=\"lazy\" class=\"\" src=\"https:\/\/biopioneer.com.tw\/wp-content\/uploads\/downloads\/2025\/06\/%E5%A4%AA%E9%BC%8E-APExBIO-Technology-LLC-%E5%93%81%E7%89%8C.png\" width=\"1099\" height=\"274\" \/><\/p>\n<p><span style=\"color: #00ccff;\"><a style=\"color: #00ccff;\" href=\"http:\/\/biopioneer.com.tw\/?p=34010\"><span style=\"text-decoration: underline; color: #33cccc;\"><strong><span style=\"font-size: 12pt;\">MS023 (type I PRMTs inhibitor\u6291\u5236\u5291) | CAS# 1831110-54-3APExBIO\u8ca8\u865f B6183<\/span><\/strong><\/span><\/a><\/span><\/p>\n<p><img decoding=\"async\" loading=\"lazy\" class=\"\" src=\"https:\/\/www.apexbt.com\/media\/diy\/images\/pathway\/epigenetics.png\" alt=\"\" width=\"933\" height=\"544\" \/><\/p>\n<p>\u8868\u89c0\u907a\u50b3\u5b78(Epigenetics)\u662f\u57fa\u56e0\u8868\u9054\u7684\u53ef\u907a\u50b3\u4fee\u98fe(heritable modifications)\uff0c\u8207 DNA \u5e8f\u5217(DNA sequence)\u7684\u8b8a\u5316\u7121\u95dc\u3002\u8868\u89c0\u907a\u50b3\u4fee\u98fe(Epigenetic modifications)\u4e3b\u8981\u767c\u751f\u5728 DNA \u6216\u7d44\u86cb\u767d\u516b\u805a\u9ad4(histone octamer)\u4e0a\u3002\u6709\u5e7e\u7a2e\u985e\u578b\u7684\u8868\u89c0\u907a\u50b3\u5b78\u4fee\u98fe(epigenetics modifications)\uff0cDNA-\u7532\u57fa\u8f49\u79fb\u9176 (DNMT) \u7684 DNA \u7532\u57fa\u5316\u548c\u7d44\u86cb\u767d\u7684\u5171\u50f9\u4fee\u98fe\uff0c\u4f8b\u5982\u4e59\u91af\u5316(acetylation)\u3001\u7532\u57fa\u5316(methylation)\u3001\u78f7\u9178\u5316(phosphorylation)\u548c\u6cdb\u7d20\u5316(ubiquitination)\u3002\u7d44\u86cb\u767d\u4e59\u91af\u8f49\u79fb\u9176 (HAT) \u7684\u7d44\u86cb\u767d\u4e59\u91af\u5316\u53c3\u8207\u8f49\u9304\u6fc0\u6d3b\uff0c\u800c\u7d44\u86cb\u767d\u53bb\u4e59\u91af\u5316\u9176 (HDAC) \u7684\u7d44\u86cb\u767d\u53bb\u4e59\u91af\u5316\u8207\u8f49\u9304\u6291\u5236(transcriptional repression)\u6709\u95dc\u3002\u7d44\u86cb\u767d\u53bb\u7532\u57fa\u5316(Histone demethylation)\u8207\u8cf4\u6c28\u9178\u7279\u7570\u6027\u53bb\u7532\u57fa\u5316\u9176 (lysine-specific demethylase , LSD) \u548c\u542b\u6709\u7d44\u86cb\u767d\u53bb\u7532\u57fa\u5316\u9176 (JHDM) \u7684 JmjC \u7d50\u69cb\u57df(JmjC domain)\u6709\u95dc\u3002<\/p>\n<p>\u6838\u5c0f\u9ad4(nucleosome)\u7531\u56db\u7a2e\u7d44\u86cb\u767d\uff08H2A\u3001H2B\u3001H3 \u548c H4\uff09\u7d44\u6210\uff0c\u5b83\u5011\u662f\u67d3\u8272\u8cea(chromatin)\u7684\u4e3b\u8981\u7d44\u6210\u90e8\u5206\u3002\u7279\u5b9a\u5316\u5b78\u57fa\u5718\u7684\u6dfb\u52a0\u548c\u53bb\u9664\u7a31\u70ba\u8868\u89c0\u907a\u50b3\u6a19\u8a18(epigenetic marks)\uff0c\u5b83\u8abf\u7bc0\u67d3\u8272\u8cea\u7d50\u69cb\u4e26\u5f71\u97ff\u57fa\u56e0\u8868\u9054\u3002\u6b64\u5916\uff0cRNA \u8207\u6291\u5236\u6027\u67d3\u8272\u8cea\u72c0\u614b(repressive chromatin state)\u7684\u5f62\u6210\u5bc6\u5207\u76f8\u95dc\u3002<\/p>\n<p>\u8868\u89c0\u907a\u50b3(Epigenetic)\u6a5f\u5236\u5728\u7d30\u80de\u6c34\u5e73\u4e0a\u97ff\u61c9\u74b0\u5883\u8b8a\u5316\uff0c\u5f9e\u800c\u5f71\u97ff\u7d30\u80de\u53ef\u5851\u6027(plasticity)\u3002\u67d3\u8272\u8cea(Chromatin)\u548c\u8868\u89c0\u907a\u50b3\u8abf\u63a7(epigenetic regulation)\u5728\u767c\u80b2\u548c\u61c9\u6fc0\u53cd\u61c9\u671f\u9593\u7684\u57fa\u56e0\u7d44\u7de8\u7a0b\u4e2d\u767c\u63ee\u91cd\u8981\u4f5c\u7528\uff0c\u8868\u89c0\u907a\u50b3\u5b78\u7f3a\u9677(defects in epigenetics)\u53ef\u5c0e\u81f4\u764c\u75c7(cancer)\u3001\u708e\u75c7(inflammation)\u548c\u4ee3\u8b1d\u7d0a\u4e82(metabolic disorders)\u7b49\u3002MG 149 \u662f\u4e00\u7a2e\u7d44\u86cb\u767d\u4e59\u91af\u8f49\u79fb\u9176 (HAT) \u6291\u5236\u5291\uff0c\u5c0d Tip60 \u548c MOF \u7684 IC50 \u503c\u5206\u5225\u70ba 74\u03bcM \u548c 47\u03bcM [1]\u3002<\/p>\n<p>MS023 is a type I PRMTs inhibitor.Protein arginine methyltransferases (PRMTs) play a critical role in various biological processes. PRMT overexpression has been observed in a variety of human diseases including cancer. PRMTs has been divided into three categories: type I PRMTs for catalyzing mono- and asymmetric dimethylation of arginine residues, type II PRMTs for catalyzing mono- and symmetric dimethylation of arginine residues, and type III PRMT for catalyzing only monomethylation of arginine residues.<\/p>\n<p><img decoding=\"async\" src=\"http:\/\/biopioneer.com.tw\/wp-content\/uploads\/2022\/09\/MS023-type-I-PRMTs-inhibitor%E6%8A%91%E5%88%B6%E5%8A%91-CAS-1831110-54-3APExBIO%E8%B2%A8%E8%99%9F-B6183-300x300.png\" alt=\"MS023 (type I PRMTs inhibitor\u6291\u5236\u5291) CAS# 1831110-54-3APExBIO\u8ca8\u865f B6183\" \/><\/p>\n<p>MS023 \u662f\u4e00\u7a2e I \u578b PRMTs \u6291\u5236\u5291\u3002\u86cb\u767d\u8cea\u7cbe\u6c28\u9178\u7532\u57fa\u8f49\u79fb\u9176 (inhibitor.Protein arginine methyltransferases ,PRMT) \u5728\u5404\u7a2e\u751f\u7269\u904e\u7a0b\u4e2d\u767c\u63ee\u8457\u95dc\u9375\u4f5c\u7528\u3002\u5df2\u5728\u5305\u62ec\u764c\u75c7(cancer)\u5728\u5167\u7684\u591a\u7a2e\u4eba\u985e\u75be\u75c5\u4e2d\u89c0\u5bdf\u5230 PRMT \u904e\u5ea6\u8868\u9054(overexpression)\u3002 PRMTs\u5206\u70ba\u4e09\u985e\uff1aI\u578bPRMTs\u7528\u65bc\u50ac\u5316\u7cbe\u6c28\u9178\u6b98\u57fa(arginine residues)\u7684\u55ae\u7532\u57fa\u5316\u548c\u4e0d\u5c0d\u7a31\u4e8c\u7532\u57fa\u5316\uff0cII\u578bPRMTs\u7528\u65bc\u50ac\u5316\u7cbe\u6c28\u9178\u6b98\u57fa(arginine residues)\u7684\u55ae\u7532\u57fa\u5316\u548c\u5c0d\u7a31\u4e8c\u7532\u57fa\u5316(symmetric demethylation)\uff0cIII\u578bPRMTs\u50c5\u50ac\u5316\u7cbe\u6c28\u9178\u6b98\u57fa\u7684\u55ae\u7532\u57fa\u5316(monomethylation)\u3002\u9ad4\u5916(In vitro)\uff1a\u5148\u524d\u7684\u7814\u7a76\u8868\u660e\uff0cMS023 \u5c0d I \u578b PRMT \u5177\u6709\u51fa\u8272\u7684\u6548\u529b\uff0c\u4f46\u5c0d II \u578b\u548c III \u578b PRMT\u3001\u86cb\u767d\u8cea\u8cf4\u6c28\u9178\u7532\u57fa\u8f49\u79fb\u9176(protein lysine methyltransferases)\u4ee5\u53ca DNA \u7532\u57fa\u8f49\u79fb\u9176(DNA methyltransferases)\u5747\u5b8c\u5168\u7121\u6d3b\u6027\u3002\u6b64\u5916\uff0cPRMT6 \u8207 MS023 \u7684\u6676\u9ad4\u7d50\u69cb\u8868\u660e MS023 \u8207\u5e95\u7269\u7d50\u5408\u4f4d\u9ede\u7d50\u5408\u3002\u6b64\u5916\uff0cMS023 \u53ef\u4ee5\u6709\u6548\u964d\u4f4e\u7d44\u86cb\u767d\u7cbe\u6c28\u9178\u4e0d\u5c0d\u7a31\u4e8c\u7532\u57fa\u5316\u7684\u7d30\u80de\u6c34\u5e73\u3002\u6b64\u5916\uff0cMS023 \u53ef\u4ee5\u964d\u4f4e\u7cbe\u6c28\u9178\u4e0d\u5c0d\u7a31\u4e8c\u7532\u57fa\u5316\u7684\u6c34\u5e73\uff0c\u540c\u6642\u9084\u53ef\u4ee5\u589e\u52a0\u7cbe\u6c28\u9178\u55ae\u7532\u57fa\u5316\u548c\u5c0d\u7a31\u4e8c\u7532\u57fa\u5316\u7684\u7d30\u80de\u6c34\u5e73 [1]\u3002\u9ad4\u5167\uff1a\u5230\u76ee\u524d\u70ba\u6b62\uff0c\u9084\u6c92\u6709\u52d5\u7269\u9ad4\u5167\u6578\u64da\u5831\u5c0e\u3002\u81e8\u5e8a\u8a66\u9a57\uff1a\u622a\u81f3\u76ee\u524d\uff0cMS023\u4ecd\u8655\u65bc\u81e8\u5e8a\u524d\u958b\u767c\u968e\u6bb5\u3002<\/p>\n<ul>\n<li>1. Pyun JH, Kim HJ, et al. &#8220;Cardiac specific PRMT1 ablation causes heart failure through CaMKII dysregulation.&#8221; Nat Commun. 2018 Nov 30;9(1):5107.\u00a0<a href=\"https:\/\/www.ncbi.nlm.nih.gov\/pubmed\/30504773\">PMID:30504773<\/a><\/li>\n<\/ul>\n<table width=\"1128\">\n<tbody>\n<tr>\n<td>Physical Appearance<\/td>\n<td>A solid<\/td>\n<\/tr>\n<tr>\n<td>Storage<\/td>\n<td>Store at -20\u00b0C<\/td>\n<\/tr>\n<tr>\n<td>M.Wt<\/td>\n<td>287.4<\/td>\n<\/tr>\n<tr>\n<td>Cas No.<\/td>\n<td>1831110-54-3<\/td>\n<\/tr>\n<tr>\n<td>Formula<\/td>\n<td>C<sub>17<\/sub>H<sub>25<\/sub>N<sub>3<\/sub>O<\/td>\n<\/tr>\n<tr>\n<td>Solubility<\/td>\n<td>\u226528.7 mg\/mL in DMSO; \u226513.7 mg\/mL in EtOH; \u226523.3 mg\/mL in H2O<\/td>\n<\/tr>\n<tr>\n<td>Chemical Name<\/td>\n<td>N1-((4-(4-isopropoxyphenyl)-1H-pyrrol-3-yl)methyl)-N1-methylethane-1,2-diamine<\/td>\n<\/tr>\n<tr>\n<td>SDF<\/td>\n<td><a href=\"https:\/\/www.apexbt.com\/downloader\/sdf\/B6183.sdf\">Download SDF<\/a><\/td>\n<\/tr>\n<tr>\n<td>Canonical SMILES<\/td>\n<td>NCCN(C)CC1=CNC=C1C2=CC=C(OC(C)C)C=C2<\/td>\n<\/tr>\n<tr>\n<td>Shipping Condition<\/td>\n<td>Ship with blue ice, or upon other requests.<\/td>\n<\/tr>\n<tr>\n<td>General tips<\/td>\n<td>For obtaining a higher solubility, please warm the tube at 37\u00b0C and shake it in the ultrasonic bath for a while. We do not recommend long-term storage for the solution, please use it up soon.<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<p>&nbsp;<\/p>\n<table width=\"553\">\n<tbody>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\">\u54c1\u9805<\/span><\/td>\n<td width=\"139\"><span style=\"color: #008080;\">CAS#<\/span><\/td>\n<td width=\"138\"><span style=\"color: #008080;\">#\u8ca8\u865f<\/span><\/td>\n<td width=\"138\"><span style=\"color: #008080;\">\u61c9\u7528<\/span><\/td>\n<\/tr>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\"><a style=\"color: #008080;\" href=\"http:\/\/biopioneer.com.tw\/?p=33999\">MG 149 \u00a0(Tip60 HAT inhibitor) \u9078\u64c7\u6027\u6291\u5236\u5291<strong><u>\u00a0<\/u><\/strong><\/a><\/span><\/td>\n<td width=\"139\"><span style=\"color: #000080;\">CAS#\u00a01243583-85-8<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">\u8ca8\u865f\u00a0B3276<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">HAT inhibitor<\/span><\/td>\n<\/tr>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\"><a style=\"color: #008080;\" href=\"http:\/\/biopioneer.com.tw\/?p=34002\">4&#8242;-bromo-Resveratrol<\/a><\/span><\/td>\n<td width=\"139\"><span style=\"color: #000080;\"><a style=\"color: #000080;\" href=\"http:\/\/biopioneer.com.tw\/?p=34002\">CAS# 1224713-90-9\u00a0<\/a><\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">\u8ca8\u865f C3552<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">Sirt1 \u548c Sirt3 \u6291\u5236\u5291<\/span><\/td>\n<\/tr>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\"><a style=\"color: #008080;\" href=\"http:\/\/biopioneer.com.tw\/?p=34010\">MS023<\/a><\/span><\/td>\n<td width=\"139\"><span style=\"color: #000080;\">CAS# 1831110-54-3<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">\u8ca8\u865f B6183<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">type I PRMTs inhibitor\u6291\u5236\u5291<\/span><\/td>\n<\/tr>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\"><a style=\"color: #008080;\" href=\"http:\/\/biopioneer.com.tw\/?p=34348\">CHZ868<\/a><\/span><\/td>\n<td width=\"139\"><span style=\"color: #000080;\">N\/O<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">\u8ca8\u865fB5980<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">Type II JAK2 inhibitor<\/span><\/td>\n<\/tr>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\"><a style=\"color: #008080;\" href=\"http:\/\/biopioneer.com.tw\/?p=35251\">Chidamide<\/a><\/span><\/td>\n<td width=\"139\"><span style=\"color: #000080;\">CAS#743420-02-2<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">\u8ca8\u865fB5916<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">Novel HDAC inhibitor<\/span><\/td>\n<\/tr>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\"><a style=\"color: #008080;\" href=\"http:\/\/biopioneer.com.tw\/?p=35254\">RGFP966<\/a><\/span><\/td>\n<td width=\"139\"><span style=\"color: #000080;\">CAS#1357389-11-7\/1396841-57-8<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">\u8ca8\u865fA8803<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">Specific HDAC3 inhibitor<\/span><\/td>\n<\/tr>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\"><a style=\"color: #008080;\" href=\"http:\/\/biopioneer.com.tw\/?p=35260\">EPZ-6438<\/a><\/span><\/td>\n<td width=\"139\"><span style=\"color: #000080;\">CAS#1403254-99-8<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">\u8ca8\u865fA8221<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">EZH2 inhibitor, potent and selective<\/span><\/td>\n<\/tr>\n<tr>\n<td width=\"139\"><span style=\"color: #008080;\"><a style=\"color: #008080;\" href=\"http:\/\/biopioneer.com.tw\/?p=35291\">Bromodomain Inhibitor, (+)-JQ1<\/a><\/span><\/td>\n<td width=\"139\"><span style=\"color: #000080;\">CAS# 1268524-70-4<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">\u8ca8\u865fA1910<\/span><\/td>\n<td width=\"138\"><span style=\"color: #000080;\">BET bromodomain inhibitor<\/span><\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<h4><\/h4>\n<p><img decoding=\"async\" loading=\"lazy\" class=\"\" src=\"http:\/\/biopioneer.com.tw\/wp-content\/uploads\/2022\/12\/%E5%93%81%E7%89%8C%E7%B9%AA%E5%9C%96-Apexbio_%E5%B7%A5%E4%BD%9C%E5%8D%80%E5%9F%9F-1-300x300.jpg\" width=\"203\" height=\"225\" \/><\/p>\n<p><a href=\"http:\/\/www.apexbt.com\/\"><span style=\"font-size: 14pt; color: #ff6600;\"><strong><span style=\"color: #800080;\"><span style=\"font-size: 14pt;\">APExBIO\u53f0\u7063\u4ee3\u7406\u5546:\u00a0 <\/span><\/span><\/strong><\/span><\/a><span style=\"font-size: 14pt;\"><a href=\"https:\/\/www.apexbt.com\/\"><span style=\"color: #ff99cc;\"><span style=\"color: #ff6600;\">https:\/\/www.apexbt.com\/<\/span><\/span><\/a><\/span><\/p>\n<p>APExBIO\u63d0\u4f9b\u512a\u8cea\u7684\u80dc\u80bd\u548c\u751f\u7269\u5206\u6790\u8a66\u5291\uff0c\u5ee3\u6cdb\u7522\u54c1\u7dda\u5982Protease\u3001Chromatin\/Epigenetics\u8868\u89c0\u907a\u50b3\u5b78\u3001MAPK Signal\u3001DNA Damege\/DNA repair\u3001\u7d30\u80de\u51cb\u4ea1\u3001\u816b\u7624\u751f\u7269\u5b78\u3001Stem cell\u7b49\u7814\u7a76\u9818\u57df\uff0c \u9084\u63d0\u4f9b\u5b9a\u5236\u7684\u670d\u52d9\uff0c\u5305\u62ec\u591a\u80bd\u5408\u6210\uff0c\u6297\u9ad4\u7684\u751f\u7522\u548c\u6aa2\u6e2c\u7684\u767c\u5c55\u3002\u7522\u54c1\u7ddaDNA\/RNA prep kit\u3001Drug Screening panel\u3001Bioactive peptides\u3001Growth factors\u3001Biotinylation Reagents\u3001tag peptides\u3001amino Acids\u3001Growth factors\u7b49\u3002APExBIO\u7522\u54c1\u8cea\u91cf\u90fd\u4f34\u96a8\u8457\u8b49\u66f8\u7684\u5206\u6790\uff0c\u9ad8\u6548\u6db2\u76f8\u8272\u8b5c\uff0c\u8cea\u8b5c\uff0c\u548cHMNR\u6578\u64da\u3002<\/p>\n<p><img decoding=\"async\" loading=\"lazy\" class=\"\" src=\"http:\/\/biopioneer.com.tw\/wp-content\/uploads\/2024\/09\/line-2_%E5%B7%A5%E4%BD%9C%E5%8D%80%E5%9F%9F-1.jpg\" width=\"302\" height=\"230\" \/><\/p>\n<table style=\"height: 2756px;\" width=\"1152\">\n<tbody>\n<tr>\n<td width=\"62\">Cat#<\/td>\n<td width=\"313\">Product Name<\/td>\n<\/tr>\n<tr>\n<td>A8743<\/td>\n<td>SYBR Safe DNA Gel Stain<\/td>\n<\/tr>\n<tr>\n<td>A6001<\/td>\n<td>3X (DYKDDDDK) Peptide<\/td>\n<\/tr>\n<tr>\n<td>K1018<\/td>\n<td>Cell Counting Kit-8 (CCK-8)<\/td>\n<\/tr>\n<tr>\n<td>A1902<\/td>\n<td>Z-VAD-FMK<\/td>\n<\/tr>\n<tr>\n<td>A3008<\/td>\n<td>Y-27632 dihydrochloride<\/td>\n<\/tr>\n<tr>\n<td>A6002<\/td>\n<td>DYKDDDDK tag Peptide<\/td>\n<\/tr>\n<tr>\n<td>B8362<\/td>\n<td>2&#8217;3&#8242;-cGAMP (sodium salt)<\/td>\n<\/tr>\n<tr>\n<td>F4002<\/td>\n<td>Phos binding reagent (Phosbind) acrylamide<\/td>\n<\/tr>\n<tr>\n<td>A8011<\/td>\n<td>Biotin-tyramide<\/td>\n<\/tr>\n<tr>\n<td>A2585<\/td>\n<td>MG-132<\/td>\n<\/tr>\n<tr>\n<td>F4005<\/td>\n<td>Prestained Protein Marker (Triple color, EDTA free, 10-250 kDa)<\/td>\n<\/tr>\n<tr>\n<td>B1274<\/td>\n<td>AP20187<\/td>\n<\/tr>\n<tr>\n<td>K1007<\/td>\n<td>Protease Inhibitor Cocktail(EDTA-Free,100X in DMSO)<\/td>\n<\/tr>\n<tr>\n<td>B8226<\/td>\n<td>InstaBlue Protein Stain Solution<\/td>\n<\/tr>\n<tr>\n<td>A3011<\/td>\n<td>CHIR-99021 (CT99021)<\/td>\n<\/tr>\n<tr>\n<td>A3007<\/td>\n<td>ABT-263 (Navitoclax)<\/td>\n<\/tr>\n<tr>\n<td>B1524<\/td>\n<td>Erastin<\/td>\n<\/tr>\n<tr>\n<td>B6055<\/td>\n<td>TCEP hydrochloride<\/td>\n<\/tr>\n<tr>\n<td>K1031<\/td>\n<td>Phusion high-fidelity DNA polymerase<\/td>\n<\/tr>\n<tr>\n<td>B1387<\/td>\n<td>(-)-Blebbistatin<\/td>\n<\/tr>\n<tr>\n<td>B4664<\/td>\n<td>T-5224<\/td>\n<\/tr>\n<tr>\n<td>A8183<\/td>\n<td>Trichostatin A (TSA)<\/td>\n<\/tr>\n<tr>\n<td>B3699<\/td>\n<td>ISRIB (trans-isomer)<\/td>\n<\/tr>\n<tr>\n<td>A1910<\/td>\n<td>Bromodomain Inhibitor, (+)-JQ1<\/td>\n<\/tr>\n<tr>\n<td>B1293<\/td>\n<td>Y-27632<\/td>\n<\/tr>\n<tr>\n<td>A8167<\/td>\n<td>Rapamycin (Sirolimus)<\/td>\n<\/tr>\n<tr>\n<td>A7024<\/td>\n<td>HOAt<\/td>\n<\/tr>\n<tr>\n<td>A7025<\/td>\n<td>HOBt (anhydrous)<\/td>\n<\/tr>\n<tr>\n<td>A8331<\/td>\n<td>Bleomycin Sulfate<\/td>\n<\/tr>\n<tr>\n<td>A4333<\/td>\n<td>CPI-613<\/td>\n<\/tr>\n<tr>\n<td>K1070<\/td>\n<td>2X SYBR Green qPCR Master Mix<\/td>\n<\/tr>\n<tr>\n<td>A8005<\/td>\n<td>Sulfo-NHS-SS-Biotin<\/td>\n<\/tr>\n<tr>\n<td>B4653<\/td>\n<td>BV6<\/td>\n<\/tr>\n<tr>\n<td>B5965<\/td>\n<td>Tamoxifen<\/td>\n<\/tr>\n<tr>\n<td>A1901<\/td>\n<td>Q-VD-OPh hydrate<\/td>\n<\/tr>\n<tr>\n<td>A8950<\/td>\n<td>UM 171<\/td>\n<\/tr>\n<tr>\n<td>K1046<\/td>\n<td>RNase Inhibitor, Murine<\/td>\n<\/tr>\n<tr>\n<td>A3317<\/td>\n<td>Clozapine N-oxide (CNO)<\/td>\n<\/tr>\n<tr>\n<td>A2614<\/td>\n<td>Bortezomib (PS-341)<\/td>\n<\/tr>\n<tr>\n<td>A8003<\/td>\n<td>Sulfo-NHS-LC-Biotin<\/td>\n<\/tr>\n<tr>\n<td>A4154<\/td>\n<td>Olaparib (AZD2281, Ku-0059436)<\/td>\n<\/tr>\n<tr>\n<td>A8012<\/td>\n<td>Biotin-XX Tyramide Reagent<\/td>\n<\/tr>\n<tr>\n<td>K1101<\/td>\n<td>PreScission Protease (PSP)<\/td>\n<\/tr>\n<tr>\n<td>A8627<\/td>\n<td>Bafilomycin A1<\/td>\n<\/tr>\n<tr>\n<td>A8001<\/td>\n<td>Sulfo-NHS-Biotin<\/td>\n<\/tr>\n<tr>\n<td>A3017<\/td>\n<td>Dasatinib (BMS-354825)<\/td>\n<\/tr>\n<tr>\n<td>A2576<\/td>\n<td>E-64<\/td>\n<\/tr>\n<tr>\n<td>K1051<\/td>\n<td>Cy3 TSA Fluorescence System Kit<\/td>\n<\/tr>\n<tr>\n<td>K1034<\/td>\n<td>2X Taq PCR Master Mix (with dye)<\/td>\n<\/tr>\n<tr>\n<td>B7972<\/td>\n<td>Pseudo-UTP<\/td>\n<\/tr>\n<tr>\n<td>A8173<\/td>\n<td>Romidepsin (FK228, depsipeptide)<\/td>\n<\/tr>\n<tr>\n<td>A4219<\/td>\n<td>Birinapant (TL32711)<\/td>\n<\/tr>\n<tr>\n<td>A4371<\/td>\n<td>Ferrostatin-1 (Fer-1)<\/td>\n<\/tr>\n<tr>\n<td>A8200<\/td>\n<td>DAPT (GSI-IX)<\/td>\n<\/tr>\n<tr>\n<td>A8249<\/td>\n<td>SB 431542<\/td>\n<\/tr>\n<tr>\n<td>K1008<\/td>\n<td>Protease Inhibitor Cocktail (EDTA-Free, 200X in DMSO)<\/td>\n<\/tr>\n<tr>\n<td>A3133<\/td>\n<td>A 83-01<\/td>\n<\/tr>\n<tr>\n<td>A8192<\/td>\n<td>Staurosporine<\/td>\n<\/tr>\n<tr>\n<td>B1054<\/td>\n<td>Resiquimod (R-848)<\/td>\n<\/tr>\n<tr>\n<td>A3018<\/td>\n<td>Trametinib (GSK1120212)<\/td>\n<\/tr>\n<tr>\n<td>A8184<\/td>\n<td>AICAR<\/td>\n<\/tr>\n<tr>\n<td>K1025<\/td>\n<td>Direct Mouse Genotyping Kit<\/td>\n<\/tr>\n<tr>\n<td>A2606<\/td>\n<td>Epoxomicin<\/td>\n<\/tr>\n<tr>\n<td>A6006<\/td>\n<td>Hexa His tag peptide<\/td>\n<\/tr>\n<tr>\n<td>A4393<\/td>\n<td>Paclitaxel (Taxol)<\/td>\n<\/tr>\n<tr>\n<td>A8315<\/td>\n<td>NU7441 (KU-57788)<\/td>\n<\/tr>\n<tr>\n<td>A4213<\/td>\n<td>Necrostatin-1<\/td>\n<\/tr>\n<tr>\n<td>A8885<\/td>\n<td>Ro 3306<\/td>\n<\/tr>\n<tr>\n<td>L1021<\/td>\n<td>DiscoveryProbe\u2122 FDA-approved Drug Library<\/td>\n<\/tr>\n<tr>\n<td>B1464<\/td>\n<td>KPT-330<\/td>\n<\/tr>\n<tr>\n<td>A8815<\/td>\n<td>SM-164<\/td>\n<\/tr>\n<tr>\n<td>B4879<\/td>\n<td>Blasticidin S HCl<\/td>\n<\/tr>\n<tr>\n<td>A8793<\/td>\n<td>N3-kethoxal<\/td>\n<\/tr>\n<tr>\n<td>K1047<\/td>\n<td>HyperScribe\u2122 T7 High Yield RNA Synthesis Kit<\/td>\n<\/tr>\n<tr>\n<td>A6004<\/td>\n<td>Influenza Hemagglutinin (HA) Peptide<\/td>\n<\/tr>\n<tr>\n<td>B1036<\/td>\n<td>MLN4924<\/td>\n<\/tr>\n<tr>\n<td>A8178<\/td>\n<td>Panobinostat (LBH589)<\/td>\n<\/tr>\n<tr>\n<td>A3963<\/td>\n<td>A-769662<\/td>\n<\/tr>\n<tr>\n<td>A3847<\/td>\n<td>SU5416<\/td>\n<\/tr>\n<tr>\n<td>B3252<\/td>\n<td>Dorsomorphin (Compound C)<\/td>\n<\/tr>\n<tr>\n<td>B4758<\/td>\n<td>BAPTA-AM<\/td>\n<\/tr>\n<tr>\n<td>A2513<\/td>\n<td>Geneticin, G-418 Sulfate<\/td>\n<\/tr>\n<tr>\n<td>B6004<\/td>\n<td>PX-478 2HCl<\/td>\n<\/tr>\n<tr>\n<td>A8955<\/td>\n<td>Z-YVAD-FMK<\/td>\n<\/tr>\n<tr>\n<td>A8193<\/td>\n<td>ABT-737<\/td>\n<\/tr>\n<tr>\n<td>B2083<\/td>\n<td>Caspofungin Acetate<\/td>\n<\/tr>\n<tr>\n<td>A8002<\/td>\n<td>NHS-Biotin<\/td>\n<\/tr>\n<tr>\n<td>A8337<\/td>\n<td>CX-5461<\/td>\n<\/tr>\n<tr>\n<td>A8312<\/td>\n<td>Torin 1<\/td>\n<\/tr>\n<tr>\n<td>A2570<\/td>\n<td>Leupeptin, Microbial<\/td>\n<\/tr>\n<tr>\n<td>K2170<\/td>\n<td>Alanine Aminotransferase (ALT or SGPT) Activity Colorimetric\/Fluorometric Assay Kit<\/td>\n<\/tr>\n<tr>\n<td>A4381<\/td>\n<td>FK866 (APO866)<\/td>\n<\/tr>\n<tr>\n<td>B2143<\/td>\n<td>Tacrolimus (FK506)<\/td>\n<\/tr>\n<tr>\n<td>A2571<\/td>\n<td>Pepstatin A<\/td>\n<\/tr>\n<tr>\n<td>k1072<\/td>\n<td>First-Strand cDNA Synthesis Kit<\/td>\n<\/tr>\n<tr>\n<td>A3003<\/td>\n<td>MDV3100 (Enzalutamide)<\/td>\n<\/tr>\n<tr>\n<td>B5997<\/td>\n<td>Dyngo-4a<\/td>\n<\/tr>\n<tr>\n<td>A3742<\/td>\n<td>Pyridostatin<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>PRMTs \u6291\u5236\u5291\u7cfb\u5217\u5546\u54c1-&gt;&gt;MS023 APExBIO Technology LLC \u662f\u4e00\u5bb6\u9818 [&hellip;]<\/p>\n","protected":false},"author":3,"featured_media":34011,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":[],"categories":[5368,486],"tags":[4930],"_links":{"self":[{"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/posts\/34010"}],"collection":[{"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/posts"}],"about":[{"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/types\/post"}],"author":[{"embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/users\/3"}],"replies":[{"embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=%2Fwp%2Fv2%2Fcomments&post=34010"}],"version-history":[{"count":5,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/posts\/34010\/revisions"}],"predecessor-version":[{"id":51903,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/posts\/34010\/revisions\/51903"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=\/wp\/v2\/media\/34011"}],"wp:attachment":[{"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=34010"}],"wp:term":[{"taxonomy":"category","embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=%2Fwp%2Fv2%2Fcategories&post=34010"},{"taxonomy":"post_tag","embeddable":true,"href":"https:\/\/biopioneer.com.tw\/index.php?rest_route=%2Fwp%2Fv2%2Ftags&post=34010"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}